Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 50042622
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50428496(CHEMBL2335204)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of sPLA2-IIA (unknown origin)-integrin alphaVbeta3 interaction in human K562 cells pretreated for 30 mins to immobilized sPLA2 before addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50428495(CHEMBL2335207)
Affinity DataIC50:  7.10E+4nMAssay Description:Inhibition of sPLA2-IIA (unknown origin)-integrin alphaVbeta3 interaction in human K562 cells pretreated for 30 mins to immobilized sPLA2 before addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50428497(CHEMBL2335203)
Affinity DataIC50:  8.50E+4nMAssay Description:Inhibition of sPLA2-IIA (unknown origin)-integrin alphaVbeta3 interaction in human K562 cells pretreated for 30 mins to immobilized sPLA2 before addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50428491(CHEMBL2335198)
Affinity DataIC50:  1.55E+5nMAssay Description:Inhibition of sPLA2-IIA (unknown origin)-integrin alphaVbeta3 interaction in human K562 cells pretreated for 30 mins to immobilized sPLA2 before addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50428492(CHEMBL2335197)
Affinity DataIC50:  2.17E+5nMAssay Description:Inhibition of sPLA2-IIA (unknown origin)-integrin alphaVbeta3 interaction in human K562 cells pretreated for 30 mins to immobilized sPLA2 before addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50428494(CHEMBL2335195)
Affinity DataIC50:  2.41E+5nMAssay Description:Inhibition of sPLA2-IIA (unknown origin)-integrin alphaVbeta3 interaction in human K562 cells pretreated for 30 mins to immobilized sPLA2 before addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50428493(CHEMBL2335196)
Affinity DataIC50:  2.62E+5nMAssay Description:Inhibition of sPLA2-IIA (unknown origin)-integrin alphaVbeta3 interaction in human K562 cells pretreated for 30 mins to immobilized sPLA2 before addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed