Compile Data Set for Download or QSAR
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Found 18 Enz. Inhib. hit(s) with all data for entry = 50005235
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489184(CHEMBL2312764)
Affinity DataIC50:  630nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489185(CHEMBL2312763)
Affinity DataIC50:  650nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489194(CHEMBL2312766)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489198(CHEMBL2312765)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489199(CHEMBL2312491)
Affinity DataIC50:  3.18E+3nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489183(CHEMBL2312770)
Affinity DataIC50:  4.67E+3nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489197(CHEMBL2312492)
Affinity DataIC50:  4.92E+3nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489200(CHEMBL2312771)
Affinity DataIC50:  5.33E+3nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489186(CHEMBL2312499)
Affinity DataIC50:  6.36E+3nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489191(CHEMBL2312496)
Affinity DataIC50:  7.01E+3nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489192(CHEMBL2312500)
Affinity DataIC50:  7.27E+3nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489187(CHEMBL2312497)
Affinity DataIC50:  1.03E+4nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489188(CHEMBL2312495)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489196(CHEMBL2312493)
Affinity DataIC50:  1.31E+4nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489195(CHEMBL2312498)
Affinity DataIC50:  1.37E+4nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489190(CHEMBL2312494)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489193(CHEMBL2312769)
Affinity DataIC50:  4.31E+4nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50489189(CHEMBL2312772)
Affinity DataIC50:  8.65E+4nMAssay Description:Inhibition of human recombinant FTase activity using dansyl-GCVLS-peptideMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed