Found 12 Enz. Inhib. hit(s) with all data for entry = 6236 
Affinity DataIC50: 1.30E+3nMAssay Description:The inhibitory potency of compounds GS4-GS8 on the 7-benzyloxy-4-(trifluoromethyl)coumarin hydroxylase activity of CYP3A4 was evaluated according to ...More data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataIC50: 2.80E+3nMAssay Description:The inhibitory potency of compounds GS4-GS8 on the 7-benzyloxy-4-(trifluoromethyl)coumarin hydroxylase activity of CYP3A4 was evaluated according to ...More data for this Ligand-Target Pair
Affinity DataIC50: 9.70E+3nMAssay Description:The inhibitory potency of compounds GS4-GS8 on the 7-benzyloxy-4-(trifluoromethyl)coumarin hydroxylase activity of CYP3A4 was evaluated according to ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:The inhibitory potency of compounds GS4-GS8 on the 7-benzyloxy-4-(trifluoromethyl)coumarin hydroxylase activity of CYP3A4 was evaluated according to ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+4nMAssay Description:The inhibitory potency of compounds GS4-GS8 on the 7-benzyloxy-4-(trifluoromethyl)coumarin hydroxylase activity of CYP3A4 was evaluated according to ...More data for this Ligand-Target Pair
Affinity DataKd: 40nMpH: 7.4Assay Description:Ligand binidng to CYP3A4 was monitored in 50 mM phosphate (pH 7.4) containing 20% glycerol and 1 mM DTT. The protein was titrated with small aliquots...More data for this Ligand-Target Pair
Affinity DataKd: 2.30E+3nMpH: 7.4Assay Description:Ligand binidng to CYP3A4 was monitored in 50 mM phosphate (pH 7.4) containing 20% glycerol and 1 mM DTT. The protein was titrated with small aliquots...More data for this Ligand-Target Pair
Affinity DataKd: 7.30E+3nMpH: 7.4Assay Description:Ligand binidng to CYP3A4 was monitored in 50 mM phosphate (pH 7.4) containing 20% glycerol and 1 mM DTT. The protein was titrated with small aliquots...More data for this Ligand-Target Pair
Affinity DataKd: 400nMpH: 7.4Assay Description:Ligand binidng to CYP3A4 was monitored in 50 mM phosphate (pH 7.4) containing 20% glycerol and 1 mM DTT. The protein was titrated with small aliquots...More data for this Ligand-Target Pair
Affinity DataKd: 1.31E+4nMpH: 7.4Assay Description:Ligand binidng to CYP3A4 was monitored in 50 mM phosphate (pH 7.4) containing 20% glycerol and 1 mM DTT. The protein was titrated with small aliquots...More data for this Ligand-Target Pair
Affinity DataKd: 160nMpH: 7.4Assay Description:Ligand binidng to CYP3A4 was monitored in 50 mM phosphate (pH 7.4) containing 20% glycerol and 1 mM DTT. The protein was titrated with small aliquots...More data for this Ligand-Target Pair
Affinity DataKd: 1.50E+3nMpH: 7.4Assay Description:Ligand binidng to CYP3A4 was monitored in 50 mM phosphate (pH 7.4) containing 20% glycerol and 1 mM DTT. The protein was titrated with small aliquots...More data for this Ligand-Target Pair
