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Found 4 Enz. Inhib. hit(s) with all data for entry = 50043291
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50438755(CHEMBL3037930)
Affinity DataKd:  30nMAssay Description:Binding affinity to XIAP BIR3-domain (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM13174((2S,4S)-1-[(2S)-3,3-dimethyl-2-[(2S)-2-(methylamin...)
Affinity DataKd:  5nMAssay Description:Binding affinity to XIAP BIR3-domain (unknown origin)More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50438757(CHEMBL2414997)
Affinity DataKd:  60nMAssay Description:Binding affinity to XIAP BIR3-domain (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM50438756(CHEMBL2414998)
Affinity DataKd:  40nMAssay Description:Binding affinity to XIAP BIR3-domain (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed