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Found 22 Enz. Inhib. hit(s) with all data for entry = 50003174
TargetAcetylcholinesterase(Mus musculus (mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM8963(CHEMBL32823 | Homodimeric Tacrine Analog 3b | N-[7...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of AChE in Swiss Webster mouse cerebral homogenate using acetylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50467895(CHEMBL4280262)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of AChE in Swiss Webster mouse cerebral homogenate using acetylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50467897(CHEMBL4287482)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of AChE in Swiss Webster mouse cerebral homogenate using acetylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50467895(CHEMBL4280262)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50467892(CHEMBL4283717)
Affinity DataIC50:  5.10nMAssay Description:Inhibition of AChE in Swiss Webster mouse cerebral homogenate using acetylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50467898(CHEMBL4282214)
Affinity DataIC50:  7.60nMAssay Description:Inhibition of AChE in Swiss Webster mouse cerebral homogenate using acetylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50467896(CHEMBL4287068)
Affinity DataIC50:  8.70nMAssay Description:Inhibition of AChE in Swiss Webster mouse cerebral homogenate using acetylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM8963(CHEMBL32823 | Homodimeric Tacrine Analog 3b | N-[7...)
Affinity DataIC50:  9.10nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50467894(CHEMBL4294287)
Affinity DataIC50:  10nMAssay Description:Inhibition of AChE in Swiss Webster mouse cerebral homogenate using acetylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50467891(CHEMBL4279148)
Affinity DataIC50:  12nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50467892(CHEMBL4283717)
Affinity DataIC50:  26nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50467898(CHEMBL4282214)
Affinity DataIC50:  26nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50467896(CHEMBL4287068)
Affinity DataIC50:  28nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50467894(CHEMBL4294287)
Affinity DataIC50:  31nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  34nMAssay Description:Inhibition of AChE in Swiss Webster mouse cerebral homogenate using acetylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
TargetCholinesterase(Mus musculus (Mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50467890(CHEMBL4290902)
Affinity DataIC50:  37nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50467897(CHEMBL4287482)
Affinity DataIC50:  37nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  63nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Mus musculus (Mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50467893(CHEMBL4276832)
Affinity DataIC50:  64nMAssay Description:Inhibition of BuChE in Swiss Webster mouse whole blood serum using butyrylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50467893(CHEMBL4276832)
Affinity DataIC50:  66nMAssay Description:Inhibition of AChE in Swiss Webster mouse cerebral homogenate using acetylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50467891(CHEMBL4279148)
Affinity DataIC50:  84nMAssay Description:Inhibition of AChE in Swiss Webster mouse cerebral homogenate using acetylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Universidade Federal Do Rio Grande Do Sul

Curated by ChEMBL
LigandPNGBDBM50467890(CHEMBL4290902)
Affinity DataIC50:  90nMAssay Description:Inhibition of AChE in Swiss Webster mouse cerebral homogenate using acetylthiocholine iodide as substrate preincubated for 10 mins followed substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed