BindingDB PrimarySearch

Found 69 Enz. Inhib. hit(s) with all data for entry = 50007549

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM220233(US9290476, 77A | US9290476, 77B | US9290476, 77C)

IC50: 3.30nMAssay Description:Inverse agonist activity at RORgammat in human PBMC derived CD4-positive T cells assessed as suppression of T cell differentiation to Th17 cells by m...More data for this Ligand-Target Pair

PDB Reactome pathway
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM220233(US9290476, 77A | US9290476, 77B | US9290476, 77C)

IC50: 3.90nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as inhibition o...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510354(CHEMBL4441287)

IC50: 5.10nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human full length RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as ...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510357(CHEMBL4543938)

IC50: 8nMAssay Description:Inverse agonist activity at RORgammat in human PBMC derived CD4-positive T cells assessed as suppression of T cell differentiation to Th17 cells by m...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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PC cid PC sid

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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510349(CHEMBL4434891)

IC50: 10nMAssay Description:Inverse agonist activity at RORgammat in human PBMC derived CD4-positive T cells assessed as suppression of T cell differentiation to Th17 cells by m...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510355(CHEMBL4552142)

IC50: 12nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as inhibition o...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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PC cid PC sid

Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510352(CHEMBL4468588)

IC50: 12nMAssay Description:Inverse agonist activity at RORgammat in human PBMC derived CD4-positive T cells assessed as suppression of T cell differentiation to Th17 cells by m...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510357(CHEMBL4543938)

IC50: 12nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human full length RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as ...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM339252(US10201546, Example 126b)

IC50: 14nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human full length RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as ...More data for this Ligand-Target Pair

PDB Reactome pathway
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3D Structure (crystal)

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM339276(US10201546, Example 136a)

IC50: 14nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as inhibition o...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM339227(US10201546, Example 112c | US10201546, Example 191...)

IC50: 17nMAssay Description:Inverse agonist activity at RORgammat in human PBMC derived CD4-positive T cells assessed as suppression of T cell differentiation to Th17 cells by m...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510352(CHEMBL4468588)

IC50: 18nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as inhibition o...More data for this Ligand-Target Pair

PDB Reactome pathway
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM339216((4-Chloro-3-((4,4-difluoropiperidin-1-yl)methyl)-2...)

IC50: 19nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as inhibition o...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM339134(US10201546, Example 68a)

IC50: 20nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as inhibition o...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM339207(US10201546, Example 103a)

IC50: 22nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as inhibition o...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510356(CHEMBL4584135)

IC50: 25nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human full length RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as ...More data for this Ligand-Target Pair

PDB Reactome pathway
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510349(CHEMBL4434891)

IC50: 29nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as inhibition o...More data for this Ligand-Target Pair

PDB Reactome pathway
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Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM339054(US10201546, Example 14a)

IC50: 30nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as inhibition o...More data for this Ligand-Target Pair

PDB Reactome pathway
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM339144(US10201546, Example 72a)

IC50: 33nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as inhibition o...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510350(CHEMBL4438967)

IC50: 41nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as inhibition o...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510347(CHEMBL4475244)

IC50: 45nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as inhibition o...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510343(CHEMBL4532727)

IC50: 50nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human full length RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as ...More data for this Ligand-Target Pair

PDB Reactome pathway
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM339227(US10201546, Example 112c | US10201546, Example 191...)

IC50: 61nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as inhibition o...More data for this Ligand-Target Pair

PDB Reactome pathway
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM220190(US9290476, 33A | US9290476, 33B | US9290476, 33C)

IC50: 95nMAssay Description:Inverse agonist activity at RORgammat in human PBMC derived CD4-positive T cells assessed as suppression of T cell differentiation to Th17 cells by m...More data for this Ligand-Target Pair

PDB Reactome pathway
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3D Structure (crystal)

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510346(CHEMBL4575356)

IC50: 116nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human full length RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as ...More data for this Ligand-Target Pair

PDB Reactome pathway
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510346(CHEMBL4575356)

IC50: 121nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as inhibition o...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510344(CHEMBL4555910)

IC50: 122nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as inhibition o...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510345(CHEMBL4517932)

IC50: 166nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human full length RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as ...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM339137(US10201546, Example 69a)

IC50: 193nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as inhibition o...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510359(CHEMBL4466031)

IC50: 280nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human full length RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as ...More data for this Ligand-Target Pair

PDB Reactome pathway
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510358(CHEMBL4459199)

IC50: 313nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human full length RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as ...More data for this Ligand-Target Pair

PDB Reactome pathway
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM339048(US10201546, Example 12a)

IC50: 327nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as inhibition o...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM339166(US10201546, Example 83)

IC50: 386nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human full length RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as ...More data for this Ligand-Target Pair

PDB Reactome pathway
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM339267(US10201546, Example 133a)

IC50: 844nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as inhibition o...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510348(CHEMBL4442831)

IC50: 2.00E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as inhibition o...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510351(CHEMBL4571921)

IC50: >6.00E+3nMAssay Description:Inverse agonist activity at GAL4-DNA binding domain-fused human RORgammat LBD expressed in pGL4.31 transfected HEK293T cells assessed as inhibition o...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM339276(US10201546, Example 136a)

Kd: 1.40nMAssay Description:Displacement of thermofluor from human recombinant N-terminal TEV cleavage site-fused-His-tagged RORgammat LBD expressed in Escherichia coli assessed...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM339144(US10201546, Example 72a)

Kd: 8.20nMAssay Description:Displacement of thermofluor from human recombinant N-terminal TEV cleavage site-fused-His-tagged RORgammat LBD expressed in Escherichia coli assessed...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510353(CHEMBL4589288)

Kd: 31nMAssay Description:Displacement of thermofluor from human recombinant N-terminal TEV cleavage site-fused-His-tagged RORgammat LBD expressed in Escherichia coli assessed...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM339137(US10201546, Example 69a)

Kd: 14nMAssay Description:Displacement of thermofluor from human recombinant N-terminal TEV cleavage site-fused-His-tagged RORgammat LBD expressed in Escherichia coli assessed...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510350(CHEMBL4438967)

Kd: 3.90nMAssay Description:Displacement of thermofluor from human recombinant N-terminal TEV cleavage site-fused-His-tagged RORgammat LBD expressed in Escherichia coli assessed...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510351(CHEMBL4571921)

Kd: 46nMAssay Description:Displacement of thermofluor from human recombinant N-terminal TEV cleavage site-fused-His-tagged RORgammat LBD expressed in Escherichia coli assessed...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM339166(US10201546, Example 83)

Kd: 357nMAssay Description:Displacement of thermofluor from human recombinant N-terminal TEV cleavage site-fused-His-tagged RORgammat LBD expressed in Escherichia coli assessed...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510354(CHEMBL4441287)

Kd: 0.0200nMAssay Description:Displacement of thermofluor from human recombinant N-terminal TEV cleavage site-fused-His-tagged RORgammat LBD expressed in Escherichia coli assessed...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510352(CHEMBL4468588)

Kd: 2.30nMAssay Description:Displacement of thermofluor from human recombinant N-terminal TEV cleavage site-fused-His-tagged RORgammat LBD expressed in Escherichia coli assessed...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510355(CHEMBL4552142)

Kd: 0.300nMAssay Description:Displacement of thermofluor from human recombinant N-terminal TEV cleavage site-fused-His-tagged RORgammat LBD expressed in Escherichia coli assessed...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510343(CHEMBL4532727)

Kd: 3.30nMAssay Description:Displacement of thermofluor from human recombinant N-terminal TEV cleavage site-fused-His-tagged RORgammat LBD expressed in Escherichia coli assessed...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510356(CHEMBL4584135)

Kd: 0.600nMAssay Description:Displacement of thermofluor from human recombinant N-terminal TEV cleavage site-fused-His-tagged RORgammat LBD expressed in Escherichia coli assessed...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM50510346(CHEMBL4575356)

Kd: 1.20nMAssay Description:Displacement of thermofluor from human recombinant N-terminal TEV cleavage site-fused-His-tagged RORgammat LBD expressed in Escherichia coli assessed...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

Nuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL

BDBM220233(US9290476, 77A | US9290476, 77B | US9290476, 77C)

Kd: 0.100nMAssay Description:Displacement of thermofluor from human recombinant N-terminal TEV cleavage site-fused-His-tagged RORgammat LBD expressed in Escherichia coli assessed...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
antibodypedia GoogleScholar

PC cid PC sid

Details Article PubMed

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