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Target
A-kinase anchor protein 7 isoform gamma
Ligand
BDBM212716
Substrate
n/a
Meas. Tech.
Binding Assay
EC50
35400±n/a nM
Citation
Tasken, K; Lygren, B; Ostensen, E; Klaveness, J Tertiary amines for use in the treatment of cardiac disorders US Patent US9951033 Publication Date 4/24/2018
More Info.:
Target
Name:
A-kinase anchor protein 7 isoform gamma
Synonyms:
A-kinase anchor protein 18 | AKA7G_MOUSE | AKAP-18 | AKAP-7 isoform gamma | Akap18 | Akap7 | PRKA7 isoform gamma | Protein kinase A-anchoring protein 7 isoform gamma
Type:
n/a
Mol. Mass.:
35486.56
Organism:
Mus musculus (Mouse)
Description:
Q7TN79
Residue:
314
Sequence:
MPFAAVDIQDDCGSPDVPQANPKRSKEEEEDRGDKNDHVKKRKKAKKDYQPNYFLSIPITNKKITTGIKVLQNSILQQDKRLTKAMVGDGSFHITLLVMQLLNEDEVNIGTDALLELKPFVEEILEGKHLALPFQGIGTFQGQVGFVKLADGDHVSALLEIAETAKRTFREKGILAGESRTFKPHLTFMKLSKAPMLRKKGVRKIEPGLYEQFIDHRFGEELLYQIDLCSMLKKKQSNGYYHCESSIVIGEKDRREPEDAELVRLSKRLVENAVLKAVQQYLEETQNKKQPGEGNSTKAEEGDRNGDGSDNNRK