Reaction Details Report a problem with these data
Target
Galanin receptor type 2
Ligand
BDBM41955
Substrate
n/a
Meas. Tech.
Dose response counterscreen for agonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for activators of beta-lactamase activity
EC50
>55700±n/a nM
Citation
 PubChem, PC Dose response counterscreen for agonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for activators of beta-lactamase activity PubChem Bioassay (2008)[AID] 
Target
Name:
Galanin receptor type 2
Synonyms:
GALNR2 | GALR2 | GALR2_HUMAN | Galanin R2 | Galanin receptor 2 | Galanin receptor type 2 | Galanin receptor type 2 (GAL2-R) (GALR2).
Type:
Enzyme Catalytic Domain
Mol. Mass.:
41724.40
Organism:
Homo sapiens (Human)
Description:
Galanin R2 GALR2 HUMAN::O43603
Residue:
387
Sequence:
MNVSGCPGAGNASQAGGGGGWHPEAVIVPLLFALIFLVGTVGNTLVLAVLLRGGQAVSTTNLFILNLGVADLCFILCCVPFQATIYTLDGWVFGSLLCKAVHFLIFLTMHASSFTLAAVSLDRYLAIRYPLHSRELRTPRNALAAIGLIWGLSLLFSGPYLSYYRQSQLANLTVCHPAWSAPRRRAMDICTFVFSYLLPVLVLGLTYARTLRYLWRAVDPVAAGSGARRAKRKVTRMILIVAALFCLCWMPHHALILCVWFGQFPLTRATYALRILSHLVSYANSCVNPIVYALVSKHFRKGFRTICAGLLGRAPGRASGRVCAAARGTHSGSVLERESSDLLHMSEAAGALRPCPGASQPCILEPCPGPSWQGPKAGDSILTVDVA
  
Inhibitor
Name:
BDBM41955
Synonyms:
5-bromanyl-2-ethoxy-N-[4-(2-methylpropylcarbamoyl)phenyl]benzamide | 5-bromo-2-ethoxy-N-[4-(2-methylpropylcarbamoyl)phenyl]benzamide | 5-bromo-2-ethoxy-N-[4-(isobutylcarbamoyl)phenyl]benzamide | 5-bromo-2-ethoxy-N-[4-[(2-methylpropylamino)-oxomethyl]phenyl]benzamide | 5-bromo-2-ethoxy-N-{4-[(isobutylamino)carbonyl]phenyl}benzamide | MLS000702062 | SMR000229312 | cid_1026561
Type:
Small organic molecule
Emp. Form.:
C20H23BrN2O3
Mol. Mass.:
419.312
SMILES:
CCOc1ccc(Br)cc1C(=O)Nc1ccc(cc1)C(=O)NCC(C)C
Structure:
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