Reaction Details Report a problem with these data
Target
Signal transducer and activator of transcription 3 [702-738,740-752]
Ligand
BDBM43602
Substrate
n/a
Meas. Tech.
Dose response cell-based assay to measure STAT3 activation
IC50
>55700±n/a nM
Citation
 PubChem, PC Dose response cell-based assay to measure STAT3 activation PubChem Bioassay (2008)[AID] 
Target
Name:
Signal transducer and activator of transcription 3 [702-738,740-752]
Synonyms:
APRF | STAT3 | STAT3_HUMAN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
5263.93
Organism:
Homo sapiens (Human)
Description:
gi_13272532
Residue:
50
Sequence:
AAPYLKTKFICVTPTTCSNTIDLPMSPRTLDSLMQFGNGEGAEPSAGGQF
  
Inhibitor
Name:
BDBM43602
Synonyms:
MLS000520930 | N-(1H-indol-3-ylmethyl)cycloheptanamine | SMR000131339 | cid_5070929 | cycloheptyl(1H-indol-3-ylmethyl)amine
Type:
Small organic molecule
Emp. Form.:
C16H22N2
Mol. Mass.:
242.3593
SMILES:
C(NC1CCCCCC1)c1c[nH]c2ccccc12
Structure:
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