Reaction Details Report a problem with these data
Target
Signal transducer and activator of transcription 3 [702-738,740-752]
Ligand
BDBM43619
Substrate
n/a
Meas. Tech.
Dose response cell-based assay to measure STAT3 activation
IC50
23520±n/a nM
Citation
 PubChem, PC Dose response cell-based assay to measure STAT3 activation PubChem Bioassay (2008)[AID] 
Target
Name:
Signal transducer and activator of transcription 3 [702-738,740-752]
Synonyms:
APRF | STAT3 | STAT3_HUMAN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
5263.93
Organism:
Homo sapiens (Human)
Description:
gi_13272532
Residue:
50
Sequence:
AAPYLKTKFICVTPTTCSNTIDLPMSPRTLDSLMQFGNGEGAEPSAGGQF
  
Inhibitor
Name:
BDBM43619
Synonyms:
2,3-dimethyl-5-(4-morpholinyl)cyclohexa-2,5-diene-1,4-dione | 2,3-dimethyl-5-morpholin-4-yl-cyclohexa-2,5-diene-1,4-dione | 2,3-dimethyl-5-morpholin-4-ylcyclohexa-2,5-diene-1,4-dione | 2,3-dimethyl-5-morpholino-p-benzoquinone | MLS000418505 | SMR000265071 | cid_2308263
Type:
Small organic molecule
Emp. Form.:
C12H15NO3
Mol. Mass.:
221.2524
SMILES:
CC1=C(C)C(=O)C(=CC1=O)N1CCOCC1 |c:1,6|
Structure:
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