Reaction Details Report a problem with these data
Target
Signal transducer and activator of transcription 3 [702-738,740-752]
Ligand
BDBM43722
Substrate
n/a
Meas. Tech.
Dose response counterscreen for STAT1 activators: cell-based high throughput assay to measure STAT3 activation
EC50
>55700±n/a nM
Citation
 PubChem, PC Dose response counterscreen for STAT1 activators: cell-based high throughput assay to measure STAT3 activation PubChem Bioassay (2008)[AID] 
Target
Name:
Signal transducer and activator of transcription 3 [702-738,740-752]
Synonyms:
APRF | STAT3 | STAT3_HUMAN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
5263.93
Organism:
Homo sapiens (Human)
Description:
gi_13272532
Residue:
50
Sequence:
AAPYLKTKFICVTPTTCSNTIDLPMSPRTLDSLMQFGNGEGAEPSAGGQF
  
Inhibitor
Name:
BDBM43722
Synonyms:
4-(5-formyl-2-furanyl)benzoic acid propyl ester | 4-(5-formyl-2-furyl)benzoic acid propyl ester | MLS000680533 | SMR000268707 | cid_1714230 | propyl 4-(5-formyl-2-furyl)benzoate | propyl 4-(5-formylfuran-2-yl)benzoate | propyl 4-(5-methanoylfuran-2-yl)benzoate
Type:
Small organic molecule
Emp. Form.:
C15H14O4
Mol. Mass.:
258.2693
SMILES:
CCCOC(=O)c1ccc(cc1)-c1ccc(C=O)o1
Structure:
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