Reaction Details Report a problem with these data
Target
Signal transducer and activator of transcription 3 [702-738,740-752]
Ligand
BDBM43739
Substrate
n/a
Meas. Tech.
Dose response counterscreen for STAT1 activators: cell-based high throughput assay to measure STAT3 activation
EC50
>55700±n/a nM
Citation
 PubChem, PC Dose response counterscreen for STAT1 activators: cell-based high throughput assay to measure STAT3 activation PubChem Bioassay (2008)[AID] 
Target
Name:
Signal transducer and activator of transcription 3 [702-738,740-752]
Synonyms:
APRF | STAT3 | STAT3_HUMAN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
5263.93
Organism:
Homo sapiens (Human)
Description:
gi_13272532
Residue:
50
Sequence:
AAPYLKTKFICVTPTTCSNTIDLPMSPRTLDSLMQFGNGEGAEPSAGGQF
  
Inhibitor
Name:
BDBM43739
Synonyms:
(2-phenylbenzotriazol-5-yl)amine | 2-phenyl-5-benzotriazolamine | 2-phenylbenzotriazol-5-amine | MLS000678352 | SMR000285263 | cid_721090
Type:
Small organic molecule
Emp. Form.:
C12H10N4
Mol. Mass.:
210.2346
SMILES:
Nc1ccc2nn(nc2c1)-c1ccccc1
Structure:
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