Reaction Details Report a problem with these data
Target
Glutathione S-transferase Mu 1
Ligand
BDBM33201
Substrate
n/a
Meas. Tech.
Profiling Assay to determine GST-GSH interactions in multiplex bead-based assays (HPSMTB buffer)
EC50
21370±n/a nM
Citation
 PubChem, PC Profiling Assay to determine GST-GSH interactions in multiplex bead-based assays (HPSMTB buffer) PubChem Bioassay (2008)[AID] 
Target
Name:
Glutathione S-transferase Mu 1
Synonyms:
GST class-mu 1 | GST1 | GSTM1 | GSTM1-1 | GSTM1_HUMAN | GSTM1a-1a | GSTM1b-1b | GTH4 | Glutathione S-transferase Mu 1 | HB subunit 4 | glutathione S-transferase
Type:
PROTEIN
Mol. Mass.:
25712.03
Organism:
Homo sapiens (Human)
Description:
ChEMBL_799596
Residue:
218
Sequence:
MPMILGYWDIRGLAHAIRLLLEYTDSSYEEKKYTMGDAPDYDRSQWLNEKFKLGLDFPNLPYLIDGAHKITQSNAILCYIARKHNLCGETEEEKIRVDILENQTMDNHMQLGMICYNPEFEKLKPKYLEELPEKLKLYSEFLGKRPWFAGNKITFVDFLVYDVLDLHRIFEPKCLDAFPNLKDFISRFEGLEKISAYMKSSRFLPRPVFSKMAVWGNK
  
Inhibitor
Name:
BDBM33201
Synonyms:
2-methyl-5,8-bis(oxidanyl)naphthalene-1,4-dione | 5,8-dihydroxy-2-methyl-1,4-naphthoquinone | 5,8-dihydroxy-2-methylnaphthalene-1,4-dione | MLS001048870 | SMR000387073 | cid_271296
Type:
Small organic molecule
Emp. Form.:
C11H8O4
Mol. Mass.:
204.1788
SMILES:
CC1=CC(=O)c2c(O)ccc(O)c2C1=O |t:1|
Structure:
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