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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM48134
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
15000±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM48134
Synonyms:
6-bromanyl-2-[(1-methylimidazol-2-yl)sulfanylmethyl]imidazo[1,2-a]pyridine | 6-bromo-2-[(1-methylimidazol-2-yl)sulfanylmethyl]imidazo[1,2-a]pyridine | 6-bromo-2-[[(1-methyl-2-imidazolyl)thio]methyl]imidazo[1,2-a]pyridine | 6-bromo-2-[[(1-methylimidazol-2-yl)thio]methyl]imidazo[1,2-a]pyridine | MLS000098102 | SMR000061182 | cid_3000090
Type:
Small organic molecule
Emp. Form.:
C12H11BrN4S
Mol. Mass.:
323.212
SMILES:
Cn1ccnc1SCc1cn2cc(Br)ccc2n1
Structure:
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