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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM48135
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
5800±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM48135
Synonyms:
5-[(4-ethoxyphenoxy)methyl]-2-furancarboxylic acid | 5-[(4-ethoxyphenoxy)methyl]-2-furoic acid | 5-[(4-ethoxyphenoxy)methyl]furan-2-carboxylic acid | MLS000043389 | SMR000020206 | cid_756954
Type:
Small organic molecule
Emp. Form.:
C14H14O5
Mol. Mass.:
262.258
SMILES:
CCOc1ccc(OCc2ccc(o2)C(O)=O)cc1
Structure:
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