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Target
DNA repair protein RAD51 homolog 1
Ligand
BDBM43853
Substrate
n/a
Meas. Tech.
Homologous recombination_Rad 51_dose response_2
IC50
53000±n/a nM
Citation
 PubChem, PC Homologous recombination_Rad 51_dose response_2 PubChem Bioassay (2008)[AID] 
Target
Name:
DNA repair protein RAD51 homolog 1
Synonyms:
RAD51 | RAD51A | RAD51_HUMAN | RECA
Type:
Enzyme Catalytic Domain
Mol. Mass.:
36960.74
Organism:
Homo sapiens (Human)
Description:
gi_49168602
Residue:
339
Sequence:
MAMQMQLEANADTSVEEESFGPQPISRLEQCGINANDVKKLEEAGFHTVEAVAYAPKKELINIKGISEAKADKILAEAAKLVPMGFTTATEFHQRRSEIIQITTGSKELDKLLQGGIETGSITEMFGEFRTGKTQICHTLAVTCQLPIDRGGGEGKAMYIDTEGTFRPERLLAVAERYGLSGSDVLDNVAYARAFNTDHQTQLLYQASAMMVESRYALLIVDSATALYRTDYSGRGELSARQMHLARFLRMLLRLADEFGVAVVITNQVVAQVDGAAMFAADPKKPIGGNIIAHASTTRLYLRKGRGETRICKIYDSPCLPEAEAMFAINADGVGDAKD
  
Inhibitor
Name:
BDBM43853
Synonyms:
3-[(4-chlorophenyl)sulfonylamino]propanoic acid [2-(4-methoxyanilino)-2-oxoethyl] ester | 3-[(4-chlorophenyl)sulfonylamino]propionic acid [2-keto-2-(p-anisidino)ethyl] ester | MLS000761252 | SMR000369563 | TL-3 | [2-(4-methoxyanilino)-2-oxoethyl] 3-[(4-chlorophenyl)sulfonylamino]propanoate | [2-[(4-methoxyphenyl)amino]-2-oxidanylidene-ethyl] 3-[(4-chlorophenyl)sulfonylamino]propanoate | cid_2122335
Type:
Small organic molecule
Emp. Form.:
C18H19ClN2O6S
Mol. Mass.:
426.871
SMILES:
COc1ccc(NC(=O)COC(=O)CCNS(=O)(=O)c2ccc(Cl)cc2)cc1
Structure:
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