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Target
POsterior Segregation
Ligand
BDBM52092
Substrate
n/a
Meas. Tech.
Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA
EC50
300000±n/a nM
Citation
 PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA PubChem Bioassay (2009)[AID] 
Target
Name:
POsterior Segregation
Synonyms:
POsterior Segregation family member (pos-1)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
29838.90
Organism:
Caenorhabditis elegans
Description:
gi_17562800
Residue:
264
Sequence:
MADNDFLSGEAIMVFKKEILDSHSDFTRSLSHQSASPEAYDQENVFSQDFQPFMKQDKETQNSASQPTSEQSLANRDPCTVPDDLREEMMRQRRKEDAFKTALCDAYKRSQACSYGDQCRFAHGVHELRLPMNPRGRNHPKYKTVLCDKFSMTGNCKYGTRCQFIHKIVDGNAAKLASGAHANTSSKSPARNAAAHNHSLFVPQGSTDRSMDLNQSLPIRQSDLVRAFARATRLDVSGYNSTAQLAQYFESQFQRIQQLSSHHH
  
Inhibitor
Name:
BDBM52092
Synonyms:
3-bromanyl-5-(3,4-dihydro-2H-quinolin-1-ylcarbonyl)pyran-2-one | 3-bromo-5-(3,4-dihydro-2H-quinoline-1-carbonyl)pyran-2-one | 3-bromo-5-[3,4-dihydro-2H-quinolin-1-yl(oxo)methyl]-2-pyranone | MLS000078343 | SMR000040194 | cid_659213
Type:
Small organic molecule
Emp. Form.:
C15H12BrNO3
Mol. Mass.:
334.165
SMILES:
Brc1cc(coc1=O)C(=O)N1CCCc2ccccc12
Structure:
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