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Target
Neuropeptide Y receptor type 2
Ligand
BDBM55926
Substrate
n/a
Meas. Tech.
Fluorescence-based cell-based high-throughput dose response assay for agonists of NPY-Y2.
EC50
>35430±n/a nM
Citation
 PubChem, PC Fluorescence-based cell-based high-throughput dose response assay for agonists of NPY-Y2. PubChem Bioassay (2009)[AID] 
Target
Name:
Neuropeptide Y receptor type 2
Synonyms:
NPY-Y2 | NPY-Y2 receptor | NPY2-R | NPY2R | NPY2R_HUMAN | Neuropeptide Y receptor type 2 | Y2 receptor | neuropeptide Y receptor Y2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42734.65
Organism:
Homo sapiens (Human)
Description:
NPY-Y2 NPY2R HUMAN::P49146
Residue:
381
Sequence:
MGPIGAEADENQTVEEMKVEQYGPQTTPRGELVPDPEPELIDSTKLIEVQVVLILAYCSIILLGVIGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGPVLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKRISFLIIGLAWGISALLASPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSIYGTVYSLSSLLILYVLPLGIISFSYTRIWSKLKNHVSPGAANDHYHQRRQKTTKMLVCVVVVFAVSWLPLHAFQLAVDIDSQVLDLKEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSVTFKAKKNLEVRKNSGPNDSFTEATNV
  
Inhibitor
Name:
BDBM55926
Synonyms:
1,5-dimethyl-4-nitro-3-pyrazolecarbothioic acid S-(4-bromophenyl) ester | 1,5-dimethyl-4-nitro-pyrazole-3-carbothioic acid S-(4-bromophenyl) ester | 4-bromophenyl 1,5-dimethyl-4-nitro-1H-pyrazole-3-carbothioate | MLS000833946 | S-(4-bromophenyl) 1,5-dimethyl-4-nitro-pyrazole-3-carbothioate | S-(4-bromophenyl) 1,5-dimethyl-4-nitropyrazole-3-carbothioate | SMR000461465 | cid_2744935
Type:
Small organic molecule
Emp. Form.:
C12H10BrN3O3S
Mol. Mass.:
356.195
SMILES:
Cc1c(c(nn1C)C(=O)Sc1ccc(Br)cc1)[N+]([O-])=O
Structure:
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