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Target
Neuropeptide Y receptor type 2
Ligand
BDBM61780
Substrate
n/a
Meas. Tech.
Fluorescence-based counterscreen for agonists of NPY-Y1: cell-based high-throughput dose response assay for agonists of NPY-Y2.
EC50
24715±n/a nM
Citation
 PubChem, PC Fluorescence-based counterscreen for agonists of NPY-Y1: cell-based high-throughput dose response assay for agonists of NPY-Y2. PubChem Bioassay (2009)[AID] 
Target
Name:
Neuropeptide Y receptor type 2
Synonyms:
NPY-Y2 | NPY-Y2 receptor | NPY2-R | NPY2R | NPY2R_HUMAN | Neuropeptide Y receptor type 2 | Y2 receptor | neuropeptide Y receptor Y2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42734.65
Organism:
Homo sapiens (Human)
Description:
NPY-Y2 NPY2R HUMAN::P49146
Residue:
381
Sequence:
MGPIGAEADENQTVEEMKVEQYGPQTTPRGELVPDPEPELIDSTKLIEVQVVLILAYCSIILLGVIGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGPVLCHLVPYAQGLAVQVSTITLTVIALDRHRCIVYHLESKISKRISFLIIGLAWGISALLASPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSIYGTVYSLSSLLILYVLPLGIISFSYTRIWSKLKNHVSPGAANDHYHQRRQKTTKMLVCVVVVFAVSWLPLHAFQLAVDIDSQVLDLKEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCEQRLDAIHSEVSVTFKAKKNLEVRKNSGPNDSFTEATNV
  
Inhibitor
Name:
BDBM61780
Synonyms:
(6E)-6-(3-salicyl-1H-benzimidazol-2-ylidene)cyclohexa-2,4-dien-1-one | (6E)-6-[3-[(2-hydroxyphenyl)methyl]-1H-benzimidazol-2-ylidene]-1-cyclohexa-2,4-dienone | (6E)-6-[3-[(2-hydroxyphenyl)methyl]-1H-benzimidazol-2-ylidene]cyclohexa-2,4-dien-1-one | 2‐{1‐[(2‐hydroxyphenyl)methyl]‐1,3‐benzodiazol‐2‐ yl}phenol (B1) | 2-[1-(2-hydroxybenzyl)-1H-benzimidazol-2-yl]phenol | MLS000060886 | SMR000069114 | cid_5392294
Type:
Small organic molecule
Emp. Form.:
C20H16N2O2
Mol. Mass.:
316.3532
SMILES:
Oc1ccccc1Cn1c(nc2ccccc12)-c1ccccc1O
Structure:
Search PDB for entries with ligand similarity: