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Target
Trans-activator protein BZLF1
Ligand
BDBM62408
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62408
Synonyms:
2-[2-Amino-1-(3-methoxy-phenyl)-4-oxo-4,5-dihydro-1H-pyrrol-3-yl]-3H-quinazolin-4-one | 2-[2-amino-4-keto-1-(3-methoxyphenyl)-2-pyrrolin-3-yl]-1H-quinazolin-4-one | 2-[5-amino-1-(3-methoxyphenyl)-3-oxo-2H-pyrrol-4-yl]-1H-quinazolin-4-one | 2-[5-azanyl-1-(3-methoxyphenyl)-3-oxidanylidene-2H-pyrrol-4-yl]-1H-quinazolin-4-one | MLS000075886 | SMR000011468 | cid_647423
Type:
Small organic molecule
Emp. Form.:
C19H16N4O3
Mol. Mass.:
348.3553
SMILES:
COc1cccc(c1)-n1cc(O)c(c1N)-c1nc2ccccc2c(=O)[nH]1
Structure:
Search PDB for entries with ligand similarity: