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Target
Trans-activator protein BZLF1
Ligand
BDBM62423
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62423
Synonyms:
1-(3-Cyano-phenyl)-3-[1-(4-methoxy-benzyl)-2-oxo-1,2-dihydro-pyridin-3-yl]-urea | 1-(3-cyanophenyl)-3-(2-keto-1-p-anisyl-3-pyridyl)urea | 1-(3-cyanophenyl)-3-[1-[(4-methoxyphenyl)methyl]-2-oxidanylidene-pyridin-3-yl]urea | 1-(3-cyanophenyl)-3-[1-[(4-methoxyphenyl)methyl]-2-oxo-3-pyridinyl]urea | 1-(3-cyanophenyl)-3-[1-[(4-methoxyphenyl)methyl]-2-oxopyridin-3-yl]urea | MLS000529619 | SMR000122094 | cid_3231725
Type:
Small organic molecule
Emp. Form.:
C21H18N4O3
Mol. Mass.:
374.3926
SMILES:
COc1ccc(Cn2cccc(NC(=O)Nc3cccc(c3)C#N)c2=O)cc1
Structure:
Search PDB for entries with ligand similarity: