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Target
Trans-activator protein BZLF1
Ligand
BDBM62448
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62448
Synonyms:
(E)-2-cyano-N-(2-furanylmethyl)-3-[1-[2-(2-methylphenoxy)ethyl]-3-indolyl]-2-propenamide | (E)-2-cyano-N-(2-furfuryl)-3-[1-[2-(2-methylphenoxy)ethyl]indol-3-yl]acrylamide | (E)-2-cyano-N-(furan-2-ylmethyl)-3-[1-[2-(2-methylphenoxy)ethyl]indol-3-yl]prop-2-enamide | 2-Cyano-N-furan-2-ylmethyl-3-[1-(2-o-tolyloxy-ethyl)-1H-indol-3-yl]-acrylamide | MLS000569137 | SMR000177626 | cid_1132164
Type:
Small organic molecule
Emp. Form.:
C26H23N3O3
Mol. Mass.:
425.4791
SMILES:
Cc1ccccc1OCCn1cc(\C=C(/C#N)C(=O)NCc2ccco2)c2ccccc12
Structure:
Search PDB for entries with ligand similarity: