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Target
Trans-activator protein BZLF1
Ligand
BDBM62501
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62501
Synonyms:
MLS001215779 | N-(5-Chloro-2-methoxy-phenyl)-2-[4-(4-fluoro-benzenesulfonyl)-piperazin-1-yl]-acetamide | N-(5-chloranyl-2-methoxy-phenyl)-2-[4-(4-fluorophenyl)sulfonylpiperazin-1-yl]ethanamide | N-(5-chloro-2-methoxy-phenyl)-2-[4-(4-fluorophenyl)sulfonylpiperazino]acetamide | N-(5-chloro-2-methoxyphenyl)-2-[4-(4-fluorophenyl)sulfonyl-1-piperazinyl]acetamide | N-(5-chloro-2-methoxyphenyl)-2-[4-(4-fluorophenyl)sulfonylpiperazin-1-yl]acetamide | SMR000613444 | cid_4797029
Type:
Small organic molecule
Emp. Form.:
C19H21ClFN3O4S
Mol. Mass.:
441.904
SMILES:
COc1ccc(Cl)cc1NC(=O)CN1CCN(CC1)S(=O)(=O)c1ccc(F)cc1
Structure:
Search PDB for entries with ligand similarity: