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Target
Trans-activator protein BZLF1
Ligand
BDBM62509
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62509
Synonyms:
MLS001160418 | N-[4-(3,4-dimethoxyphenyl)-1,2,5-oxadiazol-3-yl]-5-fluoranyl-3-methyl-1-benzofuran-2-carboxamide | N-[4-(3,4-dimethoxyphenyl)-1,2,5-oxadiazol-3-yl]-5-fluoro-3-methyl-1-benzofuran-2-carboxamide | N-[4-(3,4-dimethoxyphenyl)-1,2,5-oxadiazol-3-yl]-5-fluoro-3-methyl-2-benzofurancarboxamide | N-[4-(3,4-dimethoxyphenyl)furazan-3-yl]-5-fluoro-3-methyl-coumarilamide | SMR000652544 | cid_8035262
Type:
Small organic molecule
Emp. Form.:
C20H16FN3O5
Mol. Mass.:
397.3565
SMILES:
COc1ccc(cc1OC)-c1nonc1NC(=O)c1oc2ccc(F)cc2c1C
Structure:
Search PDB for entries with ligand similarity: