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Target
Trans-activator protein BZLF1
Ligand
BDBM62518
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62518
Synonyms:
2-(2-keto-4-methyl-chromen-7-yl)oxy-N-(4-methoxy-3-piperidinosulfonyl-phenyl)acetamide | MLS001140011 | N-(4-methoxy-3-piperidin-1-ylsulfonyl-phenyl)-2-(4-methyl-2-oxidanylidene-chromen-7-yl)oxy-ethanamide | N-(4-methoxy-3-piperidin-1-ylsulfonylphenyl)-2-(4-methyl-2-oxochromen-7-yl)oxyacetamide | N-[4-methoxy-3-(1-piperidinylsulfonyl)phenyl]-2-[(4-methyl-2-oxo-1-benzopyran-7-yl)oxy]acetamide | SMR000706009 | cid_16549413
Type:
Small organic molecule
Emp. Form.:
C24H26N2O7S
Mol. Mass.:
486.537
SMILES:
COc1ccc(NC(=O)COc2ccc3c(C)cc(=O)oc3c2)cc1S(=O)(=O)N1CCCCC1
Structure:
Search PDB for entries with ligand similarity: