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Target
Mu-type opioid receptor
Ligand
BDBM57971
Substrate
n/a
Meas. Tech.
Fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 1 (PP1)
IC50
2477±n/a nM
Citation
 PubChem, PC Fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 1 (PP1) PubChem Bioassay (2010)[AID] 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOP | MOR-1 | MOR1 | MUOR1 | Mu Opioid Receptor | Mu opiate receptor | OPIATE Mu | OPRM1 | OPRM_HUMAN | hMOP | mu-type opioid receptor isoform MOR-1
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
44789.51
Organism:
Homo sapiens (Human)
Description:
P35372
Residue:
400
Sequence:
MDSSAAPTNASNCTDALAYSSCSPAPSPGSWVNLSHLDGNLSDPCGPNRTDLGGRDSLCPPTGSPSMITAITIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKIINVCNWILSSAIGLPVMFMATTKYRQGSIDCTLTFSHPTWYWENLLKICVFIFAFIMPVLIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIHIYVIIKALVTIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSSNIEQQNSTRIRQNTRDHPSTANTVDRTNHQLENLEAETAPLP
  
Inhibitor
Name:
BDBM57971
Synonyms:
5-chloranyl-7-[piperidin-1-yl(pyridin-2-yl)methyl]quinolin-8-ol | 5-chloro-7-[1-piperidinyl(2-pyridinyl)methyl]-8-quinolinol | 5-chloro-7-[piperidin-1-yl(pyridin-2-yl)methyl]quinolin-8-ol | 5-chloro-7-[piperidino(2-pyridyl)methyl]quinolin-8-ol | MLS000774847 | SMR000365462 | cid_3491105
Type:
Small organic molecule
Emp. Form.:
C20H20ClN3O
Mol. Mass.:
353.845
SMILES:
Oc1c(cc(Cl)c2cccnc12)C(N1CCCCC1)c1ccccn1
Structure:
Search PDB for entries with ligand similarity: