Reaction Details Report a problem with these data
Target
Protein Rev
Ligand
BDBM67442
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of gld-1: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the HIV Rev protein-RRE RNA interaction
IC50
13868±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of gld-1: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the HIV Rev protein-RRE RNA interaction PubChem Bioassay (2010)[AID] 
Target
Name:
Protein Rev
Synonyms:
Human immunodeficiency virus type 1 REV | REV_HV1H2 | rev
Type:
PROTEIN
Mol. Mass.:
13078.11
Organism:
Human immunodeficiency virus 1
Description:
ChEMBL_79479
Residue:
116
Sequence:
MAGRSGDSDEELIRTVRLIKLLYQSNPPPNPEGTRQARRNRRRRWRERQRQIHSISERILGTYLGRSAEPVPLQLPPLERLTLDCNEDCGTSGTQGVGSPQILVESPTVLESGTKE
  
Inhibitor
Name:
BDBM67442
Synonyms:
3-hydroxy-1-phenalenone | 3-hydroxy-1H-phenalen-1-one | 3-hydroxyphenalen-1-one | 3-oxidanylphenalen-1-one | MLS001008607 | SMR000495845 | cid_139030
Type:
Small organic molecule
Emp. Form.:
C13H8O2
Mol. Mass.:
196.2014
SMILES:
O=C1CC(=O)c2cccc3cccc1c23
Structure:
Search PDB for entries with ligand similarity: