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Target
X-box-binding protein 1
Ligand
BDBM46553
Substrate
n/a
Meas. Tech.
XBP1 DR counterscreen for CHOP
IC50
160±n/a nM
Citation
 PubChem, PC XBP1 DR counterscreen for CHOP PubChem Bioassay (2011)[AID] 
Target
Name:
X-box-binding protein 1
Synonyms:
TREB5 | XBP1 | XBP1_HUMAN | XBP2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
28704.14
Organism:
Homo sapiens (Human)
Description:
gi_47678753
Residue:
261
Sequence:
MVVVAAAPNPADGTPKVLLLSGQPASAAGAPAGQALPLMVPAQRGASPEAASGGLPQARKRQRLTHLSPEEKALRRKLKNRVAAQTARDRKKARMSELEQQVVDLEEENQKLLLENQLLREKTHGLVVENQELRQRLGMDALVAEEEAEAKGNEVRPVAGSAESAALRLRAPLQQVQAQLSPLQNISPWILAVLTLQIQSLISCWAFWTTWTQSCSSNALPQSLPAWRSSQRSTQKDPVPYQPPFLCQWGRHQPSWKPLMN
  
Inhibitor
Name:
BDBM46553
Synonyms:
(6Z)-6-(4-anilino-6-methyl-1H-pyrimidin-2-ylidene)-1-cyclohexa-2,4-dienone | (6Z)-6-(4-anilino-6-methyl-1H-pyrimidin-2-ylidene)cyclohexa-2,4-dien-1-one | (6Z)-6-(6-methyl-4-phenylazanyl-1H-pyrimidin-2-ylidene)cyclohexa-2,4-dien-1-one | 2-(4-anilino-6-methyl-2-pyrimidinyl)phenol | MLS000062061 | SMR000070057 | cid_5413643
Type:
Small organic molecule
Emp. Form.:
C17H15N3O
Mol. Mass.:
277.3205
SMILES:
Cc1cc(Nc2ccccc2)nc(n1)-c1ccccc1O
Structure:
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