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Target
X-box-binding protein 1
Ligand
BDBM67797
Substrate
n/a
Meas. Tech.
XBP1 DR counterscreen for CHOP
IC50
7090±n/a nM
Citation
 PubChem, PC XBP1 DR counterscreen for CHOP PubChem Bioassay (2011)[AID] 
Target
Name:
X-box-binding protein 1
Synonyms:
TREB5 | XBP1 | XBP1_HUMAN | XBP2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
28704.14
Organism:
Homo sapiens (Human)
Description:
gi_47678753
Residue:
261
Sequence:
MVVVAAAPNPADGTPKVLLLSGQPASAAGAPAGQALPLMVPAQRGASPEAASGGLPQARKRQRLTHLSPEEKALRRKLKNRVAAQTARDRKKARMSELEQQVVDLEEENQKLLLENQLLREKTHGLVVENQELRQRLGMDALVAEEEAEAKGNEVRPVAGSAESAALRLRAPLQQVQAQLSPLQNISPWILAVLTLQIQSLISCWAFWTTWTQSCSSNALPQSLPAWRSSQRSTQKDPVPYQPPFLCQWGRHQPSWKPLMN
  
Inhibitor
Name:
BDBM67797
Synonyms:
5-Phenoxy-anthra[1,9-cd]isoxazol-6-one | MLS000525578 | SMR000116052 | cid_776372
Type:
Small organic molecule
Emp. Form.:
C20H11NO3
Mol. Mass.:
313.3062
SMILES:
O=C1c2ccccc2-c2onc3ccc(Oc4ccccc4)c1c23
Structure:
Search PDB for entries with ligand similarity: