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Target
Solute carrier family 22 member 2
Ligand
BDBM39344
Substrate
n/a
Meas. Tech.
ChEMBL_835924 (CHEMBL2077062)
IC50
312000±n/a nM
Citation
 Kakehi, M; Koyabu, N; Nakamura, T; Uchiumi, T; Kuwano, M; Ohtani, H; Sawada, Y Functional characterization of mouse cation transporter mOCT2 compared with mOCT1. Biochem Biophys Res Commun 296:644-50 (2002) [PubMed]  Article 
Target
Name:
Solute carrier family 22 member 2
Synonyms:
Oct2 | Organic cation transporter 2 | S22A2_MOUSE | Slc22a2
Type:
PROTEIN
Mol. Mass.:
61838.23
Organism:
Mus musculus
Description:
ChEMBL_835924
Residue:
553
Sequence:
MPTVDDILEHIGEFHLFQKQTFFLLALLSGAFTPIYVGIVFLGFTPNHHCRSPGVAELSQRCGWSPAEELNYTVPGLGSAGEVSFLSQCMRYEVDWNQSTLDCVDPLSSLAANRSHLPLSPCEHGWVYDTPGSSIVTEFNLVCAHSWMLDLFQSLVNVGFFIGAVGIGYLADRFGRKFCLLVTILINAISGVLMAISPNYAWMLVFRFLQGLVSKAGWLIGYILITEFVGLGYRRTVGICYQIAFTVGLLILAGVAYALPNWRWLQFAVTLPNFCFLLYFWCIPESPRWLISQNKNAKAMKIIKHIAKKNGKSVPVSLQSLTADEDTGMKLNPSFLDLVRTPQIRKHTLILMYNWFTSSVLYQGLIMHMGLAGDNIYLDFFYSALVEFPAAFIIILTIDRIGRRYPWAVSNMVAGAACLASVFIPDDLQWLKITVACLGRMGITIAYEMVCLVNAELYPTYIRNLAVLVCSSMCDIGGIVTPFLVYRLTDIWLEFPLVVFAVVGLVAGGLVLLLPETKGKALPETIEDAEKMQRPRKKKEKRIYLQVKKAELS
  
Inhibitor
Name:
BDBM39344
Synonyms:
4-amino-N-[2-(diethylamino)ethyl]benzamide;hydrochloride | 4-azanyl-N-[2-(diethylamino)ethyl]benzamide;hydrochloride | MLS000069436 | PROCAINAMIDE | PROCAINAMIDE HYDROCHLORIDE | SMR000059079 | cid_66068
Type:
Small organic molecule
Emp. Form.:
C13H21N3O
Mol. Mass.:
235.3253
SMILES:
CCN(CC)CCNC(=O)c1ccc(N)cc1
Structure:
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