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Target
Melanocortin receptor 4
Ligand
BDBM88496
Substrate
n/a
Meas. Tech.
Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R)
EC50
>89187±n/a nM
Citation
 PubChem, PC Luminescence-based cell-based high throughput dose response assay for biased ligands (agonists) of the melanocortin 4 receptor (MC4R) PubChem Bioassay (2012)[AID] 
Target
Name:
Melanocortin receptor 4
Synonyms:
MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R)
Type:
Enzyme
Mol. Mass.:
36949.50
Organism:
Homo sapiens (Human)
Description:
P32245
Residue:
332
Sequence:
MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLLENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVNIDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVSGILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGANMKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPLIYALRSQELRKTFKEIICCYPLGGLCDLSSRY
  
Inhibitor
Name:
BDBM88496
Synonyms:
MLS002724443 | N-(3,4-dimethylphenyl)-1-[3-[4-(1-naphthalenylmethyl)-1-piperazinyl]propyl]-1,2,4-triazole-3-carboxamide | N-(3,4-dimethylphenyl)-1-[3-[4-(1-naphthylmethyl)piperazino]propyl]-1,2,4-triazole-3-carboxamide | N-(3,4-dimethylphenyl)-1-[3-[4-(naphthalen-1-ylmethyl)piperazin-1-yl]propyl]-1,2,4-triazole-3-carboxamide | SMR001595309 | cid_45281097
Type:
Small organic molecule
Emp. Form.:
C29H34N6O
Mol. Mass.:
482.6199
SMILES:
Cc1ccc(NC(=O)c2ncn(CCCN3CCN(Cc4cccc5ccccc45)CC3)n2)cc1C
Structure:
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