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Target
Melanocortin receptor 4
Ligand
BDBM57063
Substrate
n/a
Meas. Tech.
TRFRET-based cell-based high throughput dose response assay for biased ligands (antagonists) of the melanocortin 4 receptor (MC4R)
IC50
>64564±n/a nM
Citation
 PubChem, PC TRFRET-based cell-based high throughput dose response assay for biased ligands (antagonists) of the melanocortin 4 receptor (MC4R) PubChem Bioassay (2012)[AID] 
Target
Name:
Melanocortin receptor 4
Synonyms:
MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R)
Type:
Enzyme
Mol. Mass.:
36949.50
Organism:
Homo sapiens (Human)
Description:
P32245
Residue:
332
Sequence:
MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLLENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVNIDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVSGILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGANMKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPLIYALRSQELRKTFKEIICCYPLGGLCDLSSRY
  
Inhibitor
Name:
BDBM57063
Synonyms:
1-methyl-2,4,6-triphenyl-3-propan-2-yl-4-piperidinol | 1-methyl-2,4,6-triphenyl-3-propan-2-yl-piperidin-4-ol | 1-methyl-2,4,6-triphenyl-3-propan-2-ylpiperidin-4-ol | 3-isopropyl-1-methyl-2,4,6-triphenyl-piperidin-4-ol | MLS000525447 | SMR000115921 | cid_3089037
Type:
Small organic molecule
Emp. Form.:
C27H31NO
Mol. Mass.:
385.5411
SMILES:
CC(C)C1C(N(C)C(CC1(O)c1ccccc1)c1ccccc1)c1ccccc1
Structure:
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