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Target
Melanocortin receptor 4
Ligand
BDBM88630
Substrate
n/a
Meas. Tech.
TRFRET-based cell-based high throughput dose response assay for biased ligands (antagonists) of the melanocortin 4 receptor (MC4R)
IC50
>64542±n/a nM
Citation
 PubChem, PC TRFRET-based cell-based high throughput dose response assay for biased ligands (antagonists) of the melanocortin 4 receptor (MC4R) PubChem Bioassay (2012)[AID] 
Target
Name:
Melanocortin receptor 4
Synonyms:
MC4-R | MC4R | MC4R_HUMAN | Melanocortin MC4 | Melanocortin receptor 4 (MC-4) | Melanocortin receptor 4 (MC4-R) | Melanocortin receptor 4 (MC4R)
Type:
Enzyme
Mol. Mass.:
36949.50
Organism:
Homo sapiens (Human)
Description:
P32245
Residue:
332
Sequence:
MVNSTHRGMHTSLHLWNRSSYRLHSNASESLGKGYSDGGCYEQLFVSPEVFVTLGVISLLENILVIVAIAKNKNLHSPMYFFICSLAVADMLVSVSNGSETIVITLLNSTDTDAQSFTVNIDNVIDSVICSSLLASICSLLSIAVDRYFTIFYALQYHNIMTVKRVGIIISCIWAACTVSGILFIIYSDSSAVIICLITMFFTMLALMASLYVHMFLMARLHIKRIAVLPGTGAIRQGANMKGAITLTILIGVFVVCWAPFFLHLIFYISCPQNPYCVCFMSHFNLYLILIMCNSIIDPLIYALRSQELRKTFKEIICCYPLGGLCDLSSRY
  
Inhibitor
Name:
BDBM88630
Synonyms:
6-(3-methyl-1,2,4-triazol-1-yl)-3-pyridinecarboxylic acid phenyl ester | 6-(3-methyl-1,2,4-triazol-1-yl)nicotinic acid phenyl ester | MLS000721855 | SMR000337015 | cid_1475893 | phenyl 6-(3-methyl-1,2,4-triazol-1-yl)pyridine-3-carboxylate | phenyl 6-(3-methyl-1H-1,2,4-triazol-1-yl)nicotinate
Type:
Small organic molecule
Emp. Form.:
C15H12N4O2
Mol. Mass.:
280.2814
SMILES:
Cc1ncn(n1)-c1ccc(cn1)C(=O)Oc1ccccc1
Structure:
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