Reaction Details Report a problem with these data
Target
Mitochondrial peptide methionine sulfoxide reductase
Ligand
BDBM81260
Substrate
n/a
Meas. Tech.
Absorbance-based biochemical high throughput dose response assay for activators of Methionine sulfoxide reductase A (MsrA)
EC50
>103845±n/a nM
Citation
 PubChem, PC Absorbance-based biochemical high throughput dose response assay for activators of Methionine sulfoxide reductase A (MsrA) PubChem Bioassay (2012)[AID] 
Target
Name:
Mitochondrial peptide methionine sulfoxide reductase
Synonyms:
MSRA | MSRA protein | MSRA_BOVIN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
25822.90
Organism:
Bos taurus
Description:
gi_73586699
Residue:
233
Sequence:
MLSATRRALQLFHSLFPIPRMGDSAAKIVSPQEALPGRKEPLVVAAKHHVNGNRTVEPFPEGTQMAVFGMGCFWGAERKFWTLKGVYSTQVGFAGGYTPNPTYKEVCSGKTGHAEVVRVVFQPEHISFEELLKVFWENHDPTQGMRQGNDHGSQYRSAIYPTSAEHVGAALKSKEDYQKVLSEHGFGLITTDIREGQTFYYAEDYHQQYLSKDPDGYCGLGGTGVSCPLGIKK
  
Inhibitor
Name:
BDBM81260
Synonyms:
1-methyl-4-(4-nitrobenzylidene)-2-phenyl-pyrazol[1,5-a]indol-1-ium;triflate | 1-methyl-4-[(4-nitrophenyl)methylidene]-2-phenyl-pyrazolo[1,5-a]indol-1-ium;tris(fluoranyl)methanesulfonate | 1-methyl-4-[(4-nitrophenyl)methylidene]-2-phenylpyrazolo[1,5-a]indol-1-ium;trifluoromethanesulfonate | MLS002702424 | SMR001565986 | cid_392760
Type:
Small organic molecule
Emp. Form.:
C24H18N3O2
Mol. Mass.:
380.4181
SMILES:
C[n+]1c(cc2n1c1ccccc1\c2=C/c1ccc(cc1)[N+]([O-])=O)-c1ccccc1
Structure:
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