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Target
Guanine nucleotide-binding protein subunit alpha-15
Ligand
BDBM96671
Substrate
n/a
EC50
>29904±n/a nM
Citation
 PubChem, PC Counterscreen for agonists of the human trace amine associated receptor 1 (TAAR1): Fluorescence-based cell-based high throughput dose response assay to identify nonselective Ga16 agonists PubChem Bioassay (2013)[AID] 
Target
Name:
Guanine nucleotide-binding protein subunit alpha-15
Synonyms:
G protein alpha 16 | G-protein subunit alpha-16 | G-protein subunit alpha-16 (G alpha-16) | GNA15 | GNA15_HUMAN | GNA16 | Guanine nucleotide-binding protein subunit alpha-15 [Y147C]
Type:
Protein
Mol. Mass.:
43577.62
Organism:
Homo sapiens (Human)
Description:
P30679
Residue:
374
Sequence:
MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIKQMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQDPYKVTTFEKRYAAAMQWLWRDAGIRACYERRREFHLLDSAVYYLSHLERITEEGYVPTAQDVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQCLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQGPKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVRDSVLARYLDEINLL
  
Inhibitor
Name:
BDBM96671
Synonyms:
(2-ethoxy-5-nitro-benzyl)-phenethyl-amine;hydrochloride | MLS000664875 | N-(2-ethoxy-5-nitrobenzyl)-2-phenylethanamine hydrochloride | N-[(2-ethoxy-5-nitro-phenyl)methyl]-2-phenyl-ethanamine;hydrochloride | N-[(2-ethoxy-5-nitrophenyl)methyl]-2-phenylethanamine;hydrochloride | SMR000294816 | cid_2959881
Type:
Small organic molecule
Emp. Form.:
C17H20N2O3
Mol. Mass.:
300.3523
SMILES:
CCOc1ccc(cc1CNCCc1ccccc1)[N+]([O-])=O
Structure:
Search PDB for entries with ligand similarity: