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Target
Trace amine-associated receptor 1
Ligand
BDBM96833
Substrate
n/a
EC50
5178±n/a nM
Citation
 PubChem, PC Fluorescence-based cell-based high throughput dose response assay to identify agonists of the human trace amine associated receptor 1 (TAAR1) PubChem Bioassay (2013)[AID] 
Target
Name:
Trace amine-associated receptor 1
Synonyms:
TA1 | TAAR1 | TAAR1_HUMAN | TAR1 | TRAR1 | trace amine-associated receptor 1
Type:
PROTEIN
Mol. Mass.:
39107.47
Organism:
Homo sapiens (Human)
Description:
ChEMBL_792734
Residue:
339
Sequence:
MMPFCHNIINISCVKNNWSNDVRASLYSLMVLIILTTLVGNLIVIVSISHFKQLHTPTNWLIHSMATVDFLLGCLVMPYSMVRSAEHCWYFGEVFCKIHTSTDIMLSSASIFHLSFISIDRYYAVCDPLRYKAKMNILVICVMIFISWSVPAVFAFGMIFLELNFKGAEEIYYKHVHCRGGCSVFFSKISGVLTFMTSFYIPGSIMLCVYYRIYLIAKEQARLISDANQKLQIGLEMKNGISQSKERKAVKTLGIVMGVFLICWCPFFICTVMDPFLHYIIPPTLNDVLIWFGYLNSTFNPMVYAFFYPWFRKALKMMLFGKIFQKDSSRCKLFLELSS
  
Inhibitor
Name:
BDBM96833
Synonyms:
4-[[4-[1-amino-2-(4-fluorophenyl)ethyl]-1,3-thiazol-2-yl]amino]benzenesulfonamide | 4-[[4-[1-amino-2-(4-fluorophenyl)ethyl]-2-thiazolyl]amino]benzenesulfonamide | 4-[[4-[1-amino-2-(4-fluorophenyl)ethyl]thiazol-2-yl]amino]benzenesulfonamide | 4-[[4-[1-azanyl-2-(4-fluorophenyl)ethyl]-1,3-thiazol-2-yl]amino]benzenesulfonamide | MLS003123782 | SMR001291845 | cid_46944160
Type:
Small organic molecule
Emp. Form.:
C17H17FN4O2S2
Mol. Mass.:
392.471
SMILES:
NC(Cc1ccc(F)cc1)c1csc(Nc2ccc(cc2)S(N)(=O)=O)n1
Structure:
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