Target
Guanine nucleotide-binding protein subunit alpha-15
Ligand
BDBM96917
Substrate
n/a
EC50
>29905±n/a nM
Citation
 PubChem, PC Counterscreen for antagonists of the human trace amine associated receptor 1 (TAAR1): Fluorescence-based cell-based high throughput dose reponse assay to identify nonselective Ga16 agonists PubChem Bioassay (2013)[AID] 
Target
Name:
Guanine nucleotide-binding protein subunit alpha-15
Synonyms:
G-protein subunit alpha-16 | G-protein subunit alpha-16 (G alpha-16) | GNA15 | GNA15_HUMAN | GNA16 | guanine nucleotide-binding protein subunit alpha-15
Type:
Protein
Mol. Mass.:
43577.62
Organism:
Homo sapiens (Human)
Description:
P30679
Residue:
374
Sequence:
MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIKQMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQDPYKVTTFEKRYAAAMQWLWRDAGIRAYYERRREFHLLDSAVYYLSHLERITEEGYVPTAQDVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQCLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQGPKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVRDSVLARYLDEINLL
  
Inhibitor
Name:
BDBM96917
Synonyms:
4-[(2-bromanylphenoxy)methyl]-N-pyridin-3-yl-benzamide | 4-[(2-bromophenoxy)methyl]-N-(3-pyridinyl)benzamide | 4-[(2-bromophenoxy)methyl]-N-(3-pyridyl)benzamide | 4-[(2-bromophenoxy)methyl]-N-pyridin-3-ylbenzamide | MLS001198301 | SMR000559240 | cid_1239651
Type:
Small organic molecule
Emp. Form.:
C19H15BrN2O2
Mol. Mass.:
383.239
SMILES:
Brc1ccccc1OCc1ccc(cc1)C(=O)Nc1cccnc1
Structure:
Search PDB for entries with ligand similarity: