Reaction Details
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Report a problem with these dataTarget
COUP transcription factor 2
Ligand
BDBM68101
Substrate
n/a
IC50
2663±n/a nM
Citation
PubChem, PC Luminescence-based cell-based high throughput dose response assay to identify inhibitors of COUP-TFII (NR2F2) PubChem Bioassay (2013)[AID] More Info.:
Target
Name:
COUP transcription factor 2
Synonyms:
ARP1 | COT2_HUMAN | COUP transcription factor 2 isoform a | NR2F2 | TFCOUP2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
45583.83
Organism:
Homo sapiens (Human)
Description:
gi_14149746
Residue:
414
Sequence:
MAMVVSTWRDPQDEVPGSQGSQASQAPPVPGPPPGAPHTPQTPGQGGPASTPAQTAAGGQGGPGGPGSDKQQQQQHIECVVCGDKSSGKHYGQFTCEGCKSFFKRSVRRNLSYTCRANRNCPIDQHHRNQCQYCRLKKCLKVGMRREAVQRGRMPPTQPTHGQFALTNGDPLNCHSYLSGYISLLLRAEPYPTSRFGSQCMQPNNIMGIENICELAARMLFSAVEWARNIPFFPDLQITDQVALLRLTWSELFVLNAAQCSMPLHVAPLLAAAGLHASPMSADRVVAFMDHIRIFQEQVEKLKALHVDSAEYSCLKAIVLFTSDACGLSDVAHVESLQEKSQCALEEYVRSQYPNQPTRFGKLLLRLPSLRTVSSSVIEQLFFVRLVGKTPIETLIRDMLLSGSSFNWPYMAIQ
Inhibitor
Name:
BDBM68101
Synonyms:
2-(4-tert-butylphenyl)-N'-[(Z)-2-pyrrolylidenemethyl]-1-cyclopropanecarbohydrazide | 2-(4-tert-butylphenyl)-N'-[(Z)-pyrrol-2-ylidenemethyl]cyclopropane-1-carbohydrazide | 2-(4-tert-butylphenyl)-N'-[(Z)-pyrrol-2-ylidenemethyl]cyclopropanecarbohydrazide | MLS000692856 | SMR000285625 | cid_16189574
Type:
Small organic molecule
Emp. Form.:
C19H23N3O
Mol. Mass.:
309.4054
SMILES:
CC(C)(C)c1ccc(cc1)C1CC1C(=O)NN=Cc1ccc[nH]1 |w:16.17|
Structure:
