Compile Data Set for Download or QSAR
Report error Found 6 of affinity data for UniProtKB/TrEMBL: A0A3N3ZFK4
TargetMethionine--tRNA ligase(Enterococcus faecalis)
Sun Yat-sen University

Curated by ChEMBL
LigandPNGBDBM50170723(N',N'''''-hexane-1,6-diylbis[N-(4-chlorophenyl)(im...)
Affinity DataKd:  5nMAssay Description:Binding affinity to Enterococcus faecalis type 1 MetRS expressed in Escherichia coli BL21(DE3) cells assessed as dissociation constant by ITC analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMethionine--tRNA ligase(Enterococcus faecalis)
Sun Yat-sen University

Curated by ChEMBL
LigandPNGBDBM50636199(CHEMBL5542607)
Affinity DataKd:  150nMAssay Description:Binding affinity to Enterococcus faecalis type 1 MetRS expressed in Escherichia coli BL21(DE3) cells assessed as dissociation constant in presence of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMethionine--tRNA ligase(Enterococcus faecalis)
Sun Yat-sen University

Curated by ChEMBL
LigandPNGBDBM50170723(N',N'''''-hexane-1,6-diylbis[N-(4-chlorophenyl)(im...)
Affinity DataKd:  300nMAssay Description:Binding affinity to Enterococcus faecalis type 1 MetRS expressed in Escherichia coli BL21(DE3) cells assessed as dissociation constant in presence of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMethionine--tRNA ligase(Enterococcus faecalis)
Sun Yat-sen University

Curated by ChEMBL
LigandPNGBDBM50636199(CHEMBL5542607)
Affinity DataKd:  2.70E+3nMAssay Description:Binding affinity to Enterococcus faecalis type 1 MetRS expressed in Escherichia coli BL21(DE3) cells assessed as dissociation constant by ITC analysi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMethionine--tRNA ligase(Enterococcus faecalis)
Sun Yat-sen University

Curated by ChEMBL
LigandPNGBDBM50170723(N',N'''''-hexane-1,6-diylbis[N-(4-chlorophenyl)(im...)
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of Enterococcus faecalis type 1 MetRS expressed in Escherichia coli BL21(DE3) cells measured after 1.5 hrs in presence of ATP by pre-trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetMethionine--tRNA ligase(Enterococcus faecalis)
Sun Yat-sen University

Curated by ChEMBL
LigandPNGBDBM50636199(CHEMBL5542607)
Affinity DataIC50: 1.61E+4nMAssay Description:Inhibition of Enterococcus faecalis type 1 MetRS expressed in Escherichia coli BL21(DE3) cells measured after 1.5 hrs in presence of ATP by pre-trans...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed