Compile Data Set for Download or QSAR
Report error Found 189 of affinity data for UniProtKB/TrEMBL: O08590
TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309489BDBM309489(US9603833, Example 111)
Affinity DataIC50: 0.400nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228079BDBM228079(US9556160, ex 126)
Affinity DataIC50: 0.530nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309497BDBM309497(US9603833, Example 120)
Affinity DataIC50: 0.600nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309490BDBM309490(US9603833, Example 112)
Affinity DataIC50: 0.700nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309491BDBM309491(US9603833, Example 113)
Affinity DataIC50: 0.700nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309479BDBM309479(US9603833, Example 92)
Affinity DataIC50: 0.800nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309486BDBM309486(US9603833, Example 108)
Affinity DataIC50: 0.800nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228098BDBM228098(US9556160, ex 559 | US9556160, ex 567)
Affinity DataIC50: 0.810nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228098BDBM228098(US9556160, ex 559 | US9556160, ex 567)
Affinity DataIC50: 0.810nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309476BDBM309476(US9603833, Example 88)
Affinity DataIC50: 0.900nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309477BDBM309477(US9603833, Example 89)
Affinity DataIC50: 0.900nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228087BDBM228087(US9556160, ex 316)
Affinity DataIC50: 0.900nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228083BDBM228083(US9556160, ex 273)
Affinity DataIC50: 0.950nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228093BDBM228093(US9556160, ex 554)
Affinity DataIC50: 0.970nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228084BDBM228084(US9556160, ex 293)
Affinity DataIC50: 0.970nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309474BDBM309474(US9603833, Example 86)
Affinity DataIC50: 1nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228082BDBM228082(US9556160, ex 220)
Affinity DataIC50: 1nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228072BDBM228072(US9556160, ex 63)
Affinity DataIC50: 1.10nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309459BDBM309459(US9603833, Example 12)
Affinity DataIC50: 1.10nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309464BDBM309464(US9603833, Example 45)
Affinity DataIC50: 1.20nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309492BDBM309492(US9603833, Example 114)
Affinity DataIC50: 1.20nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228097BDBM228097(US9556160, ex 558)
Affinity DataIC50: 1.20nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228105BDBM228105(US9556160, ex 566)
Affinity DataIC50: 1.20nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309470BDBM309470(US9603833, Example 70)
Affinity DataIC50: 1.30nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228095BDBM228095(US9556160, ex 556)
Affinity DataIC50: 1.30nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309487BDBM309487(US9603833, Example 109)
Affinity DataIC50: 1.40nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228077BDBM228077(US9556160, ex 110)
Affinity DataIC50: 1.40nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228101BDBM228101(US9556160, ex 562)
Affinity DataIC50: 1.40nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228099BDBM228099(US9556160, ex 560)
Affinity DataIC50: 1.40nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309475BDBM309475(US9603833, Example 87)
Affinity DataIC50: 1.40nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309478BDBM309478(US9603833, Example 90)
Affinity DataIC50: 1.40nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228102BDBM228102(US9556160, ex 563)
Affinity DataIC50: 1.5nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228103BDBM228103(US9556160, ex 564)
Affinity DataIC50: 1.5nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309488BDBM309488(US9603833, Example 110)
Affinity DataIC50: 1.60nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228100BDBM228100(US9556160, ex 561)
Affinity DataIC50: 1.60nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309498BDBM309498(US9603833, Example 121)
Affinity DataIC50: 1.60nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228096BDBM228096(US9556160, ex 557)
Affinity DataIC50: 1.60nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228078BDBM228078(US9556160, ex 118)
Affinity DataIC50: 1.70nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228085BDBM228085(US9556160, ex 300)
Affinity DataIC50: 1.70nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 50184850BDBM50184850(N'-[2-(4-fluorophenyl)allyl]-N-methylhydrazine hyd...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of SSAO in rat lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228071BDBM228071(US9556160, ex 52)
Affinity DataIC50: 1.70nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228090BDBM228090(US9556160, ex 551)
Affinity DataIC50: 1.80nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228073BDBM228073(US9556160, ex 74)
Affinity DataIC50: 1.80nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228070BDBM228070(US9556160, ex 29)
Affinity DataIC50: 1.90nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309473BDBM309473(US9603833, Example 85)
Affinity DataIC50: 1.90nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228075BDBM228075(US9556160, ex 83)
Affinity DataIC50: 1.90nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 50184849BDBM50184849(N'-(2-phenylallyl)hydrazine hydrochloride | CHEMBL...)
Affinity DataIC50: 2nMAssay Description:Inhibition of SSAO in rat lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228089BDBM228089(US9556160, ex 335)
Affinity DataIC50: 2nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 309482BDBM309482(US9603833, Example 101)
Affinity DataIC50: 2.10nMAssay Description:The compounds of the present invention obtained in Production Examples were examined for the inhibitory effect on human and rat VAP-1 enzyme (SSAO) b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetMembrane primary amine oxidase(Rat)
R-Tech Ueno

US Patent
LigandChemical structure of BindingDB Monomer ID 228080BDBM228080(US9556160, ex 157)
Affinity DataIC50: 2.10nMT: 2°CAssay Description:A rat VAP-1 enzyme (SSAO) (reference: Biol Pharm Bull. 2005 March; 28(3): 413-8) activity was measured by a radiochemistry-enzymatic assay using 14C-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2018
Entry Details
US Patent

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