Compile Data Set for Download or QSAR
Report error Found 394 of affinity data for UniProtKB/TrEMBL: O14578
LigandPNGBDBM50643185(CHEMBL5572737 | US20250243196, Compound F-90)
Affinity DataKd:  0.300nMAssay Description:Binding affinity to NanoLuc fused-CITK kinase domain (unknown origin) expressed in HEK293T cells assessed as dissociation constant NanoBRET Target En...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM130909(US8822500, Stauro- sporine | US9920060, Staurospor...)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of human STK21 using KKRPQRRYSNVF as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition and measured after 120 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM761568((2R)-2-Amino-N-[4-[2-(difluoromethyl)-1H-pyrrolo[2...)
Affinity DataIC50: 4nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643144(CHEMBL5595104 | US20250243196, Compound F-9)
Affinity DataIC50: 4.90nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643187(CHEMBL5591534 | US20250243196, Compound F-162)
Affinity DataIC50: 5nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643187(CHEMBL5591534 | US20250243196, Compound F-162)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM761490((2R)-2-Amino-4,4-dimethyl-N-[3-methyl-4-(1H-pyrrol...)
Affinity DataIC50: 7.80nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643161(CHEMBL5569359 | US20250243196, Compound F-58)
Affinity DataIC50: 8.10nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM761575((2R)-2-Amino-N-[6-[2-(difluoromethyl)-1H-pyrrolo[2...)
Affinity DataIC50: 9nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM761482((2R)-2-Amino-4,4-dimethyl-N-[4-(2-methyl-1H-pyrrol...)
Affinity DataIC50: 9.10nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643185(CHEMBL5572737 | US20250243196, Compound F-90)
Affinity DataKd:  9.5nMAssay Description:Binding affinity to NanoLuc fused-CITK (unknown origin) expressed in HEK293T cells assessed as dissociation constant NanoBRET Target Engagement Intra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM761581((2R)-2-Amino-N-[2-fluoro-3-methyl-4-(2-methyl-1H-p...)
Affinity DataIC50: 10nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM761566((2R)-2-Amino-N-[4-(2-cyclopropyl-1H-pyrrolo[2,3-b]...)
Affinity DataIC50: 10nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643156(CHEMBL5568742 | US20250243196, Compound F-21)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643156(CHEMBL5568742 | US20250243196, Compound F-21)
Affinity DataIC50: 10.4nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM761532((2R)-2-Amino-N-[4-[2-(difluoromethyl)-1H-pyrrolo[2...)
Affinity DataIC50: 11.7nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643185(CHEMBL5572737 | US20250243196, Compound F-90)
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643185(CHEMBL5572737 | US20250243196, Compound F-90)
Affinity DataIC50: 12nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643144(CHEMBL5595104 | US20250243196, Compound F-9)
Affinity DataIC50: 12.5nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM15138(Biochemistry 469551 Compound 11 | 5-indazolyl pyri...)
Affinity DataKd:  13nMAssay Description:Binding constant for CIT kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
LigandPNGBDBM50643144(CHEMBL5595104 | US20250243196, Compound F-9)
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643157(CHEMBL5575901 | US20250243196, Compound F-16)
Affinity DataIC50: 13.8nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643157(CHEMBL5575901 | US20250243196, Compound F-16)
Affinity DataIC50: 14nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM761442(2-Amino-4,4-dimethyl-N-[4-(1H-pyrrolo[2,3-b]pyridi...)
Affinity DataIC50: 14.1nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643161(CHEMBL5569359 | US20250243196, Compound F-58)
Affinity DataIC50: 15nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643136(CHEMBL5579704 | US20250243196, Compound F-13)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643188(CHEMBL5575300 | US20250243196, Compound F-161)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643136(CHEMBL5579704 | US20250243196, Compound F-13)
Affinity DataIC50: 16.6nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643183(CHEMBL5595678 | US20250243196, Compound F-57)
Affinity DataIC50: 16.8nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643183(CHEMBL5595678 | US20250243196, Compound F-57)
Affinity DataIC50: 17nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM761502((2R)-2-Amino-N-[2-fluoro-3-methyl-4-(1H-pyrrolo[2,...)
Affinity DataIC50: 17nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643164(CHEMBL5590268 | US20250243196, Compound F-62)
Affinity DataIC50: 17nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643164(CHEMBL5590268 | US20250243196, Compound F-62)
Affinity DataIC50: 17.1nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643184(CHEMBL5575657 | US20250243196, Compound F-89)
Affinity DataIC50: 18nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM761567((2R)-2-Amino-N-[4-(2-cyclopropyl-1H-pyrrolo[2,3-b]...)
Affinity DataIC50: 18nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM761573((2R)-2-Amino-N-[2-methoxy-6-(2-methyl-1H-pyrrolo[2...)
Affinity DataIC50: 18nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM761531((2R)-2-Amino-N-[4-[2-(difluoromethyl)-1H-pyrrolo[2...)
Affinity DataIC50: 18.1nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643184(CHEMBL5575657 | US20250243196, Compound F-89)
Affinity DataIC50: 18.8nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643188(CHEMBL5575300 | US20250243196, Compound F-161)
Affinity DataIC50: 19nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643136(CHEMBL5579704 | US20250243196, Compound F-13)
Affinity DataIC50: 19.6nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643180(CHEMBL5574799 | US20250243196, Compound F-48)
Affinity DataIC50: 20nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643146(CHEMBL5566667 | US20250243196, Compound F-41)
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant CITK kinase domain assessed as phosphorylation of substrate ULight-ARTKQTARKSTGGKAPRICQLAGC measured after 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM761512((R)-2-Amino-N-(3-(difluoromethoxy)-4-(1H-pyrrolo[2...)
Affinity DataIC50: 21.5nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643180(CHEMBL5574799 | US20250243196, Compound F-48)
Affinity DataIC50: 21.9nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM761569((2R)-2-amino-4,4-dimethyl-N-[4-[2-(trifluoromethyl...)
Affinity DataIC50: 22nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643146(CHEMBL5566667 | US20250243196, Compound F-41)
Affinity DataIC50: 22.1nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM761562((2R)-2-Amino-N-[2-fluoro-3-methyl-4-(1H-pyrrolo[2,...)
Affinity DataIC50: 23.1nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM50643138(CHEMBL5571250 | US20250243196, Compound F-33)
Affinity DataIC50: 23.8nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM761572((2R)-2-Amino-N-[2-fluoro-3-methyl-4-[2-(trifluorom...)
Affinity DataIC50: 24nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM761570((2R)-2-Amino-4,4-dimethyl-N-(6-(2-methyl-1H-pyrrol...)
Affinity DataIC50: 26nMAssay Description:TBDMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

Displayed 1 to 50 (of 394 total ) | Next | Last >>
Jump to: