Compile Data Set for Download or QSAR
Report error Found 19 for UniProtKB: O77240
TargetEcdysone receptor/Protein ultraspiracle homolog(Spruce budworm moth)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  0.501nMAssay Description:Binding affinity to Choristoneura fumiferana EcRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Spruce budworm moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128305(N'-tert-butyl-N'-(3,5-dimethylbenzoyl)-3-methoxy-2...)
Affinity DataEC50:  280nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Spruce budworm moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128297(5-Ethyl-2,3-dihydro-benzo[1,4]dioxine-6-carboxylic...)
Affinity DataEC50:  390nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Spruce budworm moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128309(3,5-Dimethyl-benzoic acid N-tert-butyl-N'-(2-ethyl...)
Affinity DataEC50:  410nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Spruce budworm moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128312(3-Methoxy-N-[1-(2-methoxy-benzoyl)-cyclohexyl]-2-m...)
Affinity DataEC50:  1.03E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Spruce budworm moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128300(N-[1-(3,5-Dimethyl-benzoyl)-cyclohexyl]-3-methoxy-...)
Affinity DataEC50:  1.11E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Spruce budworm moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128302(N-[1-(3,5-Dimethyl-benzoyl)-cyclohexyl]-2-ethyl-3-...)
Affinity DataEC50:  1.25E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Spruce budworm moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128304(N-[4-(3,5-Dimethyl-benzoyl)-tetrahydro-thiopyran-4...)
Affinity DataEC50:  1.80E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Spruce budworm moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128313(N-[1-(3,5-Dimethyl-benzoyl)-cyclopentyl]-3-methoxy...)
Affinity DataEC50:  1.91E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Spruce budworm moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128315(N-[1-(3,5-Dimethyl-benzoyl)-cycloheptyl]-3-methoxy...)
Affinity DataEC50:  2.97E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Spruce budworm moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128299(4-Methyl-benzo[1,3]dioxole-5-carboxylic acid [1-(3...)
Affinity DataEC50:  3.22E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Spruce budworm moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128306(3-Methoxy-N-[1-(2-methoxy-benzoyl)-cycloheptyl]-2-...)
Affinity DataEC50:  3.36E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Spruce budworm moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128298(N-[1-(3,5-Dimethyl-benzoyl)-1-ethyl-propyl]-3-meth...)
Affinity DataEC50:  6.23E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Spruce budworm moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128303(3-Methoxy-N-[1-(2-methoxy-benzoyl)-cyclopentyl]-2-...)
Affinity DataEC50:  6.61E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Spruce budworm moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128301(N-[1-(3,5-Dimethyl-benzoyl)-cyclobutyl]-3-methoxy-...)
Affinity DataEC50:  1.00E+4nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Spruce budworm moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128307(N-[4-(3,5-Dimethyl-benzoyl)-tetrahydro-pyran-4-yl]...)
Affinity DataEC50:  1.00E+4nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Spruce budworm moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128308(N-[4-(3,5-Dimethyl-benzoyl)-1,1-dioxo-hexahydro-1l...)
Affinity DataEC50:  3.00E+4nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Spruce budworm moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128310(N-[1-(3,5-Dimethyl-benzoyl)-cyclopropyl]-3-methoxy...)
Affinity DataEC50:  3.33E+4nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Spruce budworm moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128311(N-[2-(3,5-Dimethyl-phenyl)-1,1-dimethyl-2-oxo-ethy...)
Affinity DataEC50:  4.20E+4nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Choristoneura fumiferana (CfEcR) and a luciferase reporter gene in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed