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Report error Found 118 of affinity data for UniProtKB/TrEMBL: P12955
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50366413(PHOSPHOENOLPYRUVATE)
Affinity DataKi:  8.5nMpH: 6.0Assay Description:Inhibition of prolidase from swine kidney at a pH 6More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285931(2-((1R,2R)-2-Carboxy-cyclopentyl)-2-oxo-ethyl-ammo...)
Affinity DataKi:  270nMAssay Description:Inhibitory activity against porcine kidney prolidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632022(CHEMBL5419166)
Affinity DataIC50: 280nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632026(CHEMBL5433567)
Affinity DataIC50: 290nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632008(CHEMBL5435351)
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50366413(PHOSPHOENOLPYRUVATE)
Affinity DataKi:  300nMAssay Description:Inhibitory constant for inhibition of prolidase in the first phase of biphasic inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50368352(Cerubidine | DAUNORUBICIN)
Affinity DataIC50: 300nMAssay Description:Inhibition of prolidase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632007(CHEMBL5429139)
Affinity DataIC50: 530nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  547nMAssay Description:Binding affinity to human PEPD incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632037(CHEMBL5433668)
Affinity DataIC50: 560nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50078402((S)-1-((R)-3-Amino-2-hydroxy-5-methyl-hexanoyl)-py...)
Affinity DataIC50: 660nMAssay Description:Inhibition against Prolidase from pig kidney.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632002(CHEMBL5437413)
Affinity DataIC50: 670nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632038(CHEMBL5393876)
Affinity DataIC50: 720nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632029(CHEMBL5419034)
Affinity DataIC50: 720nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632031(CHEMBL5401781)
Affinity DataIC50: 840nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632015(CHEMBL5407130)
Affinity DataIC50: 840nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632030(CHEMBL5410658)
Affinity DataIC50: 910nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632016(CHEMBL5403940)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632028(CHEMBL5399924)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632004(CHEMBL5396150)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632005(CHEMBL5438777)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632034(CHEMBL5436435)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632024(CHEMBL5396773)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632012(CHEMBL5398054)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632013(CHEMBL5421036)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632006(CHEMBL5394915)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632014(CHEMBL5404330)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50078394((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition against Prolidase from pig kidney.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632017(CHEMBL5433606)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50078397(1-(3-Amino-2-hydroxy-5-methyl-hexanoyl)-pyrrolidin...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition against Prolidase from pig kidney.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632011(CHEMBL5406619)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632039(CHEMBL5419938)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632033(CHEMBL5430934)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632010(CHEMBL5403929)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50078401((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition against Prolidase from pig kidney.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632040(CHEMBL5400780)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632025(CHEMBL5432938)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632032(CHEMBL5403523)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632041(CHEMBL5438224)
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50632003(CHEMBL5403681)
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of recombinant human PEPD using Ala-Pro as substrate assessed as alanine release by measuring increase in fluorescense signal by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50645729(CHEMBL5592090)
Affinity DataKi:  9.73E+3nMAssay Description:Competitive inhibition of prolidase (unknown origin) in erythrocytes assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50232504((2R)-4-[5,8-dimethyl-3-(trifluoromethyl)-5,6-dihyd...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50232518((2R)-4-oxo-4-[8-(pyridin-2-ylmethyl)-3-(trifluorom...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50232518((2R)-4-oxo-4-[8-(pyridin-2-ylmethyl)-3-(trifluorom...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50232510((2R)-4-[8-benzyl-3-(trifluoromethyl)-5,6-dihydro[1...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50232519((2R)-4-[8-[3,5-bis(trifluoromethyl)benzyl]-3-(trif...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50232505((2R)-4-[5,5-dimethyl-3-(trifluoromethyl)-5,6-dihyd...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50232507(2-[7-[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50232510((2R)-4-[8-benzyl-3-(trifluoromethyl)-5,6-dihydro[1...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
TargetXaa-Pro dipeptidase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50232514((2R)-4-[8-allyl-3-(trifluoromethyl)-5,6-dihydro[[1...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2012
Entry Details Article
PubMed
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