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Report error Found 97 for UniProtKB: P17538
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50073139([2,2-dimethyl-3-(N-(4-cyanobenzoyl)aminoi)-5-pheny...)
Affinity DataIC50: 2.10nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075109(1,1-dimethyl-2-phenylcarboxamidoheptanoic anhydrid...)
Affinity DataIC50: 5.30nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50024092(6-Iodomethylene-4-phenyl-tetrahydro-pyran-2-one | ...)
Affinity DataKi:  5.30nMAssay Description:Binding constant alpha-chymotrypsin was determined by competitive inhibition assay with Suc-Ala-Ala-Pro-Phe-pNA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50142284(2-Ethyl-1,1-dioxo-1,2,3,4,6,7-hexahydro-5,8-dioxa-...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against chymotrypsinogen; Range 1-10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2012
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075107(1,1-dimethyl-4-phenyl-2-propylcarboxamidopentanoic...)
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075107(1,1-dimethyl-4-phenyl-2-propylcarboxamidopentanoic...)
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075110(2-(4-cyanophenylcarboxamido)-1,1-dimethyl-2-phenyl...)
Affinity DataIC50: 15nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50014743(CHEMBL132171 | N-(1-{2-[2-(1-Benzyl-3,3,3-trifluor...)
Affinity DataKi:  17nMAssay Description:Binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075106(1,1-dimethyl-4-phenyl-2-phenylcarboxamidopentanoic...)
Affinity DataIC50: 18nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075106(1,1-dimethyl-4-phenyl-2-phenylcarboxamidopentanoic...)
Affinity DataIC50: 18nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075114(1,1-dimethyl-2-phenylcarboxamidooctanoic anhydride...)
Affinity DataIC50: 31nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075104(1,1-dimethyl-2-phenylcarboxamidononanoic anhydride...)
Affinity DataIC50: 44nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075118(1,1-dimethyl-2-phenylcarboxamidohexanoic anhydride...)
Affinity DataIC50: 49nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50289952(6-Dimethylamino-5-methyl-2-(1-phenyl-ethylamino)-b...)
Affinity DataIC50: 65nMAssay Description:Inhibitory concentration against human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075105(1,1-dimethyl-2-phenylcarboxamidopentanoic anhydrid...)
Affinity DataIC50: 72nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50014731(CHEMBL130006 | 3-[(1-{2-[2-(3-Methoxycarbonyl-prop...)
Affinity DataKi:  79nMAssay Description:Binding affinity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50289954(5-Methyl-2-(1-phenyl-ethylamino)-benzo[d][1,3]oxaz...)
Affinity DataIC50: 88nMAssay Description:Inhibitory concentration against human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075113(1,1-dimethyl-2-phenylcarboxamidopropanoic anhydrid...)
Affinity DataIC50: 140nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50289953(2-[1-(4-Bromo-phenyl)-ethylamino]-5-methyl-benzo[d...)
Affinity DataIC50: 140nMAssay Description:Inhibitory concentration against human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50289955(5-Methyl-2-(1-phenyl-ethylamino)-benzo[d][1,3]oxaz...)
Affinity DataIC50: 180nMAssay Description:Inhibitory concentration against human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075116(2-(4-cyanophenylcarboxamido)-1,1-dimethyl-2-(2-met...)
Affinity DataIC50: 190nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075111(2-(4-cyanophenylcarboxamido)-2-cyclohex-3-enyl-1,1...)
Affinity DataIC50: 220nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075108(2-(2-chlorophenyl)-2-(4-cyanophenylcarboxamido)-1,...)
Affinity DataIC50: 250nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50025866(N-[1R-(2-phenyl ethyl)]benzamide difluoroborane | ...)
Affinity DataKi:  270nMAssay Description:Competitive inhibition of alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50025877(N-[1R-(2-phenyl ethyl)]propanamide difluoroborane ...)
Affinity DataKi:  290nMAssay Description:Competitive inhibition of alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50069989(CHEMBL325041 | (R)-3-methyl-1-((S)-3-phenyl-2-(pyr...)
Affinity DataKi:  320nMAssay Description:Inhibitory activity against human ChymotrypsinogenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50025875(2-Amino-N-[1R-(2-phenyl ethyl)]propanamide boronic...)
Affinity DataKi:  320nMAssay Description:Competitive inhibition of alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50025872(N-[1R-(2-phenyl ethyl)]benzamide boronic acid | CH...)
Affinity DataKi:  360nMAssay Description:Competitive inhibition of alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM521743(US11149067, Compound Ahp2)
Affinity DataKi:  370nMAssay Description:In general, proteolytic activity was tested by monitoring the cleavage of the specific chromogenic substrate at 405 nm wavelength for 60 or 120 minut...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2022
Entry Details
US Patent

TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50025860(N-(2-phenyl ethyl)benzamide boronic acid | CHEMBL2...)
Affinity DataKi:  650nMAssay Description:Competitive inhibition of alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50025870(N-(2-phenyl ethyl)benzamide difluoroborane | CHEMB...)
Affinity DataKi:  650nMAssay Description:Competitive inhibition of alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50070440({(S)-1-[(S)-1-(1-Benzylcarbamoyl-4-oxo-azetidin-2-...)
Affinity DataIC50: 800nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075112(1,1-dimethyl-2-propylcarboxamidooctanoic anhydride...)
Affinity DataIC50: 810nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50025868(2-Amino-N-(2-phenyl ethyl)propanamide difluorobora...)
Affinity DataKi:  1.40E+3nMAssay Description:Competitive inhibition of alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50025865(N-[1R-(2-phenyl ethyl)]acetamide difluoroborane | ...)
Affinity DataKi:  1.70E+3nMAssay Description:Competitive inhibition of alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50070444((3R,4S)-3-Methyl-2-oxo-4-(pyridin-2-ylmethylsulfan...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50063719(2-Isopropylamino-5-methyl-benzo[d][1,3]oxazin-4-on...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory concentration against human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50025874(2-Amino-N-benzylpropanamide difluoroborane | CHEMB...)
Affinity DataKi:  2.00E+3nMAssay Description:Competitive inhibition of alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50025862(N-[1R-(2-phenyl ethyl)]acetamide boronic acid | CH...)
Affinity DataKi:  2.10E+3nMAssay Description:Competitive inhibition of alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM521750(US11149067, Compound Ahp9)
Affinity DataKi:  2.10E+3nMAssay Description:In general, proteolytic activity was tested by monitoring the cleavage of the specific chromogenic substrate at 405 nm wavelength for 60 or 120 minut...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2022
Entry Details
US Patent

TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50289948(2-Dimethylamino-N-[5-methyl-4-oxo-2-(1-phenyl-ethy...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibitory concentration against human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50289950(4-Methoxy-N-[5-methyl-4-oxo-2-(1-phenyl-ethylamino...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibitory concentration against human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50139465(((S)-1-Mercaptomethyl-2-phenyl-ethyl)-carbamic aci...)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibitory activity against chymotrypsinogen in the presence of Zn(II) (500 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50133629(2,3-Dioxo-2,3-dihydro-indole-1-carboxylic acid ben...)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition constant against alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075117(2-phenylcarboxamidopropanoic anhydride | CHEMBL134...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50025861(N-benzylbenzamide difluoroborane | CHEMBL56829)
Affinity DataKi:  5.00E+3nMAssay Description:Competitive inhibition of alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50139460(((R)-1-Mercaptomethyl-2-phenyl-ethyl)-carbamic aci...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory activity against chymotrypsinogen in the presence of Zn(II) (500 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50025859(N-(2-phenyl ethyl)acetamide boronic acid | CHEMBL6...)
Affinity DataKi:  6.50E+3nMAssay Description:Competitive inhibition of alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50025863(2-Amino-N-[(1R)-benzyl]propanamide difluoroborane ...)
Affinity DataKi:  6.50E+3nMAssay Description:Competitive inhibition of alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50025871(N-(2-phenyl ethyl)acetamide difluoroborane | CHEMB...)
Affinity DataKi:  7.40E+3nMAssay Description:Competitive inhibition of alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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