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Report error Found 126 of affinity data for UniProtKB/TrEMBL: P19367
TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169033(CHEMBL3806069)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169038(CHEMBL3804841)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169026(CHEMBL3805148)
Affinity DataIC50:  16nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169032(CHEMBL3805398)
Affinity DataIC50:  20nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169037(CHEMBL3805205)
Affinity DataIC50:  20nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169034(CHEMBL3805734)
Affinity DataIC50:  25nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169031(CHEMBL3805905)
Affinity DataIC50:  32nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169017(CHEMBL3804930)
Affinity DataIC50:  40nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169028(CHEMBL3805598)
Affinity DataIC50:  160nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169023(CHEMBL3805753)
Affinity DataIC50:  160nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169015(CHEMBL3805460)
Affinity DataIC50:  790nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169042(CHEMBL3806103)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169036(CHEMBL3806028)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169039(CHEMBL3806132)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169019(CHEMBL3805765)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169013(CHEMBL3805703)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169025(CHEMBL3806250)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169041(CHEMBL3805653)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169040(CHEMBL3804874)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169014(CHEMBL3806183)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169043(CHEMBL3806095)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169046(CHEMBL3805459)
Affinity DataIC50:  6.30E+4nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169018(CHEMBL3804924)
Affinity DataIC50:  1.60E+5nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169020(CHEMBL3805806)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169022(CHEMBL3805752)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM32004(2-(3-Oxo-1,3-dihydro-indol-2-ylidene)-indan-1,3-di...)
Affinity DataEC50:  3.71E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM80764(MLS000031522 | N-[2-[4-(2-hydroxyethyl)-1-piperazi...)
Affinity DataEC50:  2.40E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM80765(8-(3,4-dimethoxyphenyl)-1,3-dimethyl-7-[(3-phenyl-...)
Affinity DataEC50:  3.51E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM80766(2-(7-fluoro-2-methyl-4-thiazolo[5,4-b]indolyl)acet...)
Affinity DataEC50:  8.10E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM34343(4-(6-ethylindolo[2,3-b]quinoxalin-2-yl)sulfonylmor...)
Affinity DataEC50: >8.00E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM80767(1-[2-(3,4-dihydro-1H-isoquinolin-2-yl)-2-keto-ethy...)
Affinity DataEC50:  3.67E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM80768(1-[2-(1-azepanyl)-2-oxoethyl]-8-methyl-4-[1]benzop...)
Affinity DataEC50:  2.17E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM42405(MLS000110376 | N-(2-piperazin-1-yl-1,2-dihydroacen...)
Affinity DataEC50:  1.36E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM34648((4-chlorodithiazol-5-ylidene)-(4,6-dimethyl-2-pyri...)
Affinity DataEC50:  3.99E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM80769(1-[(4-chlorobenzylidene)amino]-2-imino-3-(4-methyl...)
Affinity DataEC50: >8.00E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM80770(4-(3-bromophenyl)-1,3-thiazol-2-amine | 4-(3-bromo...)
Affinity DataEC50:  4.93E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM48647(2-[[2-[[1-(4-methoxyphenyl)-5-tetrazolyl]thio]-1-o...)
Affinity DataEC50:  3.74E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM46685((4-chlorodithiazol-5-ylidene)-(p-tolyl)amine | 4-c...)
Affinity DataEC50:  5.32E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM80773((3-chlorophenyl)-[5-(2,3-dihydro-1,4-benzodioxin-6...)
Affinity DataEC50:  4.13E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM48288(MLS000565792 | N-ethyl-5-(4-methylphenyl)-6H-1,3,4...)
Affinity DataEC50:  6.31E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM80774(5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-(4-methoxyp...)
Affinity DataEC50:  2.39E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM80775(1-[4-(4-tert-butylphenyl)-1,3-thiazol-2-yl]-2-(3,4...)
Affinity DataEC50:  4.74E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM74476(4-({[1-(4-chlorophenyl)-3-methyl-5-oxo-1,5-dihydro...)
Affinity DataEC50: >8.00E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM80776(2-Acetylamino-5-benzyl-4-methyl-thiophene-3-carbox...)
Affinity DataEC50:  3.94E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM80777((6E)-6-[[(4-amino-1,2,4-triazol-3-yl)hydrazo]methy...)
Affinity DataEC50:  4.23E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM65111((4E)-5-methyl-2-phenyl-4-[[(5-phenyl-1,2,4-triazin...)
Affinity DataEC50: >8.00E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM67197(1,1-dibutyl-3-[[(Z)-(3-methyl-5-oxidanylidene-1-ph...)
Affinity DataEC50: >8.00E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM80778(3-(2-ketochromen-3-yl)-N-(4-pyrrolidinophenyl)benz...)
Affinity DataEC50: >8.00E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM47735(3-chloranyl-N-(3,3-dimethylbutan-2-yl)-6-nitro-1-b...)
Affinity DataEC50:  4.68E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

TargetHexokinase-1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM80779(MLS000547762 | N-[2-(4-Methyl-4H-[1,2,4]triazol-3-...)
Affinity DataEC50:  2.47E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay

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