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Report error Found 2288 of affinity data for UniProtKB/TrEMBL: P29371
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432251(CHEMBL2347505)
Affinity DataEC50:  0.00540nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432272(CHEMBL2347491)
Affinity DataEC50:  0.0120nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50299467((5S,8S,14S,17S,20S,23S,26S,29S,32S)-26-((1H-imidaz...)
Affinity DataEC50:  0.0130nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432243(CHEMBL2347513)
Affinity DataEC50:  0.0170nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432246(CHEMBL2347510)
Affinity DataEC50:  0.0240nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432244(CHEMBL2347512)
Affinity DataEC50:  0.0260nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432267(CHEMBL2347496)
Affinity DataEC50:  0.0320nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432265(CHEMBL2347498)
Affinity DataEC50:  0.0360nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432271(CHEMBL2347492)
Affinity DataEC50:  0.0360nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432248(CHEMBL2347508)
Affinity DataEC50:  0.0380nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432247(CHEMBL2347509)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432269(CHEMBL2347494)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432266(CHEMBL2347497)
Affinity DataEC50:  0.0410nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432270(CHEMBL2347493)
Affinity DataEC50:  0.0430nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432268(CHEMBL2347495)
Affinity DataEC50:  0.0460nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432274(CHEMBL2347489)
Affinity DataEC50:  0.0510nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432273(CHEMBL2347490)
Affinity DataEC50:  0.0600nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432275(CHEMBL2347488)
Affinity DataEC50:  0.0650nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432250(CHEMBL2347506)
Affinity DataEC50:  0.0710nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432242(CHEMBL2347361)
Affinity DataEC50:  0.0720nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432259(CHEMBL2347662)
Affinity DataEC50:  0.0780nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432264(CHEMBL2347657)
Affinity DataEC50:  0.0790nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432245(CHEMBL2347511)
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432262(CHEMBL2347659)
Affinity DataEC50:  0.0830nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432258(CHEMBL2347499)
Affinity DataEC50:  0.0850nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432256(CHEMBL2347501)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432261(UPEROLEIN)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432260(CHEMBL2347661)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432254(CHEMBL2347502)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50291261(SR-14280 | SR-142801 | (S)-(+)-N-((3-[1-Benzoyl-3-...)
Affinity DataKd:  0.200nMAssay Description:Equilibrium binding affinity to human NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50291261(SR-14280 | SR-142801 | (S)-(+)-N-((3-[1-Benzoyl-3-...)
Affinity DataKd:  0.200nMAssay Description:Binding affinity to wild type human NK3 receptor expressed in HEK293 cells assessed as [3H]IP accumulation after 45 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50291261(SR-14280 | SR-142801 | (S)-(+)-N-((3-[1-Benzoyl-3-...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to NK3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50281562(Asp-Val-Pro-Lys-Ser-Asp-Gln-Phe-Val-Gly-Leu-Met-NH...)
Affinity DataEC50:  0.210nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50051290(SR 142806 | CHEMBL299377 | SR 142801 | N-(1-{3-[1-...)
Affinity DataKi:  0.210nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2011
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50051290(SR 142806 | CHEMBL299377 | SR 142801 | N-(1-{3-[1-...)
Affinity DataKi:  0.210nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2011
Entry Details
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50291261(SR-14280 | SR-142801 | (S)-(+)-N-((3-[1-Benzoyl-3-...)
Affinity DataIC50: 0.210nMAssay Description:Compound was tested for binding affinity against human Tachykinin receptor 3 in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50194558(CHEMBL373569 | ELEDOISIN)
Affinity DataEC50:  0.220nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50291261(SR-14280 | SR-142801 | (S)-(+)-N-((3-[1-Benzoyl-3-...)
Affinity DataKd:  0.220nMAssay Description:Apparent binding affinity to human NK3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50432241(CHEMBL2347362)
Affinity DataEC50:  0.280nMAssay Description:Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50299467((5S,8S,14S,17S,20S,23S,26S,29S,32S)-26-((1H-imidaz...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to human NK3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50116722(N-{(R)-5-{4-[3-((R)-1-Carbamoyl-2-hydroxy-ethyl)-2...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity against recombinant human tachykinin receptor 3 in CHO cells using [125I][MePhe]-NKB as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM233239(US9346786, 43)
Affinity DataKi:  0.300nM ΔG°:  -50.5kJ/molepH: 7.4 T: 2°CAssay Description:hNK3 receptor binding experiment were performed using [3H]SR142801 (Catalog No. TRK1035, specific activity: 74.0 Ci/mmol, Amersham, GE Healthcare UK ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2017
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50116736(N-{(R)-5-{4-[3-(1-Carbamoyl-1-methyl-ethyl)-2-oxo-...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity against recombinant human tachykinin receptor 3 in CHO cells using [125I][MePhe]-NKB as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50116078(CHEMBL66332 | SCH 206272 | 3,5-Dichloro-N-[3-(3,4-...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50116717(3,5-Dichloro-N-[(R)-3-(3,4-dichloro-phenyl)-2-[(Z)...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity against recombinant human tachykinin receptor 3 in CHO cells using [125I][MePhe]-NKB as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50505284(CHEMBL4576324)
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I][MePhe]NKB from human NK3 receptor expressed in CHO cells membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM85083(NKB [MePhe7])
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2012
Entry Details
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM85083(NKB [MePhe7])
Affinity DataKi:  0.340nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50445820(CHEMBL3104783)
Affinity DataKi:  0.398nMAssay Description:Displacement of [3H]-SR142801 from human NK3 receptor expressed in recombinant CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetNeuromedin-K receptor(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50116745(N-{(R)-5-[4-(3-Carbamoylmethyl-2-oxo-tetrahydro-py...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity against recombinant human tachykinin receptor 3 in CHO cells using [125I][MePhe]-NKB as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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