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Report error Found 718 of affinity data for UniProtKB/TrEMBL: P30411
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50413782(CHEMBL1627325)
Affinity DataEC50:  0.0339nMAssay Description:Antagonist activity at human recombinant bradykinin 2 receptor expressed in CHO cells assessed as inhibition of bradykinin-induced intracellular calc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419921(CHEMBL1956864)
Affinity DataKi:  0.0398nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50049949(2-(2-{[1-(2-{2-[2-({1-[1-(2-Amino-5-guanidino-pent...)
Affinity DataEC50:  0.0490nMAssay Description:Antagonist activity at human recombinant bradykinin 2 receptor expressed in CHO cells assessed as inhibition of bradykinin-induced intracellular calc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50293905((S)-4-amino-5-(4-(4-(2,4-dichloro-3-((2,4-dimethyl...)
Affinity DataIC50: 0.0500nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419920(CHEMBL1956863)
Affinity DataKi:  0.0501nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419924(CHEMBL1956856)
Affinity DataKi:  0.0501nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419907(CHEMBL1956855)
Affinity DataKi:  0.0501nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50411275(MEN-16132 | CHEMBL218427)
Affinity DataKi:  0.0501nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419899(CHEMBL1956876)
Affinity DataKi:  0.0501nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50411275(MEN-16132 | CHEMBL218427)
Affinity DataKd:  0.0501nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50403371(Firazyr | HOE-140 | ICATIBANT)
Affinity DataKi:  0.0600nMAssay Description:Binding affinity towards human cloned Bradykinin receptor B2 expressed in CHO cells by [3H]bradykinin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419909(CHEMBL1956858)
Affinity DataKi:  0.0631nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419922(CHEMBL1956870)
Affinity DataKi:  0.0631nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419918(CHEMBL1956719)
Affinity DataKi:  0.0631nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50403371(Firazyr | HOE-140 | ICATIBANT)
Affinity DataKi:  0.0640nMAssay Description:Binding affinity against human cloned Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50049949(2-(2-{[1-(2-{2-[2-({1-[1-(2-Amino-5-guanidino-pent...)
Affinity DataKi:  0.0650nMAssay Description:Binding affinity towards human cloned Bradykinin receptor B2 expressed in CHO cells by [3H]bradykinin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50081659((3-(Ser-Thi-Gly-Hyp-Pro-Arg-Lys-H)-4-oxo-3,4-dihyd...)
Affinity DataKi:  0.0700nMAssay Description:Binding affinity towards human cloned Bradykinin receptor B2 expressed in CHO cells by [3H]bradykinin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419913(CHEMBL1956862)
Affinity DataKi:  0.0794nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419901(CHEMBL1956720)
Affinity DataKi:  0.0794nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419902(CHEMBL1956722)
Affinity DataKi:  0.0794nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419906(CHEMBL1956854)
Affinity DataKi:  0.0794nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50089308(H-DArg-Arg-Pro-Hyp-Gly-Thi-Ser-DTic-Oic-Arg-OH( HO...)
Affinity DataKi:  0.0800nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50403371(Firazyr | HOE-140 | ICATIBANT)
Affinity DataIC50: 0.0900nMAssay Description:In vitro inhibitory activity towards bradykinin receptor B2 using [3H]BK (0.06 nM) as a radioligand in guinea pig ileum membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50403371(Firazyr | HOE-140 | ICATIBANT)
Affinity DataIC50: 0.0900nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50403371(Firazyr | HOE-140 | ICATIBANT)
Affinity DataIC50: 0.0900nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50146108(Arg-Arg-Pro-Hyp-Gly-Thi-Cys-Tic-Oic-Arg | CHEMBL27...)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419912(CHEMBL1956861)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419908(CHEMBL1956857)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419905(CHEMBL1956853)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50049949(2-(2-{[1-(2-{2-[2-({1-[1-(2-Amino-5-guanidino-pent...)
Affinity DataKi:  0.110nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419924(CHEMBL1956856)
Affinity DataKd:  0.123nMAssay Description:Antagonist activity at human bradykinin B2 receptor expressed in dhfr-deficient CHO cells assessed as inhibition of bradykinin-induced inositol monop...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419900(CHEMBL1956718)
Affinity DataKi:  0.126nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419919(CHEMBL1956721)
Affinity DataKi:  0.126nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419903(CHEMBL1956723)
Affinity DataKi:  0.126nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50067317(N-({[2,4-Dichloro-3-(2-methyl-quinolin-8-yloxymeth...)
Affinity DataIC50: 0.130nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/8/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50052513(8-Methyl-3-(2-oxo-propyl)-1-phenethyl-1,3,8-triaza...)
Affinity DataKi:  0.150nMAssay Description:Affinity to human Bradykinin receptor B2 in CHO cell membranes determined by displacement of [3H]-NPC 17731More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419898(CHEMBL1956875)
Affinity DataKi:  0.158nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50142956(4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-pyrazol-1-...)
Affinity DataIC50: 0.170nMAssay Description:In vitro inhibitory activity towards human bradykinin receptor B2 expressed in CHO cells using [3H]BK (1.0 nM) as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50142944(4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-pyrazol-1-...)
Affinity DataIC50: 0.180nMAssay Description:In vitro inhibitory activity towards human bradykinin receptor B2 expressed in CHO cells using [3H]BK (1.0 nM) as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50614474(CHEMBL5274928)
Affinity DataKi:  0.180nMAssay Description:Binding affinity to B2 bradykinin receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50146893(4-{(E)-2-[({[2,4-Dichloro-3-(4-ethoxy-2-methyl-qui...)
Affinity DataIC50: 0.190nMAssay Description:Concentration required to inhibit specific binding of [3H]-BK(0.06 nM) to the bradykinin receptor B2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419904(CHEMBL1956852)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419897(CHEMBL1955876)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50146905(4-{(E)-2-[({[2,4-Dichloro-3-(4-methoxy-2-methyl-qu...)
Affinity DataIC50: 0.230nMAssay Description:Concentration required to inhibit specific binding of [3H]-BK(0.06 nM) to the bradykinin receptor B2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50142952(4-{(E)-2-[({[2,4-Dichloro-3-(2-methyl-4-[1,2,4]tri...)
Affinity DataIC50: 0.230nMAssay Description:In vitro inhibitory activity towards human bradykinin receptor B2 expressed in CHO cells using [3H]BK (1.0 nM) as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50142951(4-[3-({[2,4-Dichloro-3-(4-imidazol-1-yl-2-methyl-q...)
Affinity DataIC50: 0.230nMAssay Description:In vitro inhibitory activity towards human bradykinin receptor B2 expressed in CHO cells using [3H]BK (1.0 nM) as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419911(CHEMBL1956860)
Affinity DataKi:  0.251nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419910(CHEMBL1956859)
Affinity DataKi:  0.251nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50419917(CHEMBL1956867)
Affinity DataKi:  0.251nMAssay Description:Displacement of [3H]-Bradykinin from human bradykinin B2 receptor expressed in CHO cells membrane after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Human)
National Institute of Neuroscienc

Curated by ChEMBL
LigandPNGBDBM50142954(4-[(E)-2-({1-[2,4-Dichloro-3-(4-imidazol-1-yl-2-me...)
Affinity DataIC50: 0.260nMAssay Description:Displacement of [3H]bradykinin from human recombinant bradykinin B2 receptor expressed in CHO cells incubated for 2 hrs by liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
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