Compile Data Set for Download or QSAR
Report error Found 1586 for UniProtKB: P30551
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089269(N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[3-(1H-indol-3...)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061828(N-(1-Carbamoyl-2-phenyl-ethyl)-3-({2-[3-(1H-indol-...)
Affinity DataKi:  0.0300nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061829((R)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-({(S)-2-[...)
Affinity DataKi:  0.0300nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061828(N-(1-Carbamoyl-2-phenyl-ethyl)-3-({2-[3-(1H-indol-...)
Affinity DataKi:  0.0300nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50003666(3-[2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 0.0500nMAssay Description:Inhibitory activity against cholecystokinin type A receptor from rat pancreas binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50003669(CHEMBL411079 | Ac-Tyr(SO3H)-Met-Gly-Trp-Met-R-Dtc-...)
Affinity DataIC50: 0.0500nMAssay Description:Concentration inhibiting [3H]propionyl-CCK-8 binding to cholecystokinin type A receptor of rat pancreatic membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50089268(N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2-[2-(2-{2-[2-(4...)
Affinity DataKi:  0.0500nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061832((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-{(S)-2-[(...)
Affinity DataKi:  0.0700nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.0794nMAssay Description:Binding affinity against cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.0800nMAssay Description:Half maximal inhibition of specific binding of [125I]-Bolton-Hunter CCK-8 to Cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.0800nMAssay Description:Displacement of [125 I] CCK-8 from Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of [125I]Cholecystokinin-8 (125I-CCK-8) binding to Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article
PDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of binding of [125I]- CCK-33 to rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.0800nMAssay Description:Half-maximal inhibition of [125I]CCK-33 binding to cholecystokinin A receptor from rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.0800nMAssay Description:The compound was tested for its activity to inhibit the binding of [3H]-L-364,718 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article
PDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.0800nMAssay Description:Concentration required for 50% inhibition of Cholecystokinin type A receptor in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.0800nMAssay Description:Ability to inhibit the binding of [125I]CCK-8 to Cholecystokinin type A receptor in rat pancreas.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article
PDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.0900nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50170765([(S)-1-((4aS,5R)-2-Benzyl-1-mercapto-3-oxo-octahyd...)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of 71 pM [125I]BH-(Thr,Nle)CCK-9 binding to rat cholecystokinin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50106593([1-(2-Benzyl-3-oxo-1-thioxo-octahydro-4a(S)-pyrido...)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of [3H]pCCK-8 binding to cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.0900nMAssay Description:Inhibition of [125I]BH-CCK-8 binding to Cholecystokinin type A receptor of rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50170765([(S)-1-((4aS,5R)-2-Benzyl-1-mercapto-3-oxo-octahyd...)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of 71 pM [125I]BH-(Thr,Nle)CCK-9 binding to rat cholecystokinin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50: 0.100nMAssay Description:Evaluated for inhibition of CCK-A receptor by displacing [125I]bolton hunter CCK-8 radioligand in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50033600(Asp-Tyr(SO3H)-Met-Gly-Trp-Met-Asp-Phe-NH2 | CHEMBL...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of binding of [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreas.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.100nMAssay Description:Half-maximal inhibition of specific binding of [125I]bolton hunter CCK-8 to rat pancreas cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50281617(Asp Tyr (OSO3H) Met Gly Trp Met Asp Phe | CHEMBL26...)
Affinity DataIC50: 0.100nMAssay Description:Compound was tested for the inhibition of specific binding of [125I]bolton Hunter CCK-8 to Cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of binding of [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreas.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article
PDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of binding of [125I]Bolton-Hunter labeled CCK-8 to cholecystokinin type A receptor in the rat pancreas.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50: 0.100nMAssay Description:Half-maximal inhibition of specific binding of [125I]bolton hunter CCK-8 to rat pancreas cholecystokinin type A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataKi:  0.148nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM81962(S-L-365,260)
Affinity DataKi:  0.148nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50449787(PD-134308 | CHEMBL2062154)
Affinity DataKi:  0.148nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50023142(1H-Indole-2-carboxylic acid [6-(2-fluoro-phenyl)-1...)
Affinity DataIC50: 0.200nMAssay Description:Displacement of [125I]CCK from Cholecystokinin receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50061833((R)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-{(S)-2-[(...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50026690(2-[2-(2-{2-[2-{2-[2-(2-Amino-3-phenyl-propionylami...)
Affinity DataIC50: 0.200nMAssay Description:Compound was tested for in vitro inhibition of the binding of [125I](Nle11)-HG-13 to Histamine H2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50369326(CHEMBL1791002)
Affinity DataKi:  0.240nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50011545(CHEMBL430906 | Desamino-Tyr(SO3H)-Met-Gly-Trp-Met-...)
Affinity DataIC50: 0.25nMAssay Description:Inhibition of [3H]propanoyl binding to cholecystokinin type A receptor was determined in fresh rat pancreatic tissue membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50456295(CHEMBL2111920)
Affinity DataIC50: 0.260nMAssay Description:Inhibition of binding of [125I]CCK-8 to cholecystokinin type A receptor in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of [125I]- Bolton-Hunter CCK-26-33 binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50060321(CHEMBL419764 | 1H-Indole-2-carboxylic acid (1-meth...)
Affinity DataKi:  0.300nMAssay Description:Inhibition of [3H]pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50367648(CHEMBL1907661)
Affinity DataIC50: 0.300nMAssay Description:Half-maximal inhibition of [125I]CCK-8 binding to cholecystokinin receptor from rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50281730(4-Chloro-N-((S)-1-methyl-2-oxo-5-phenyl-2,3-dihydr...)
Affinity DataIC50: 0.390nMAssay Description:The compound was tested for its activity to inhibit the binding of [3H]-L-364,718 to Cholecystokinin type A receptor in rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50367623(CHEMBL1907852)
Affinity DataIC50: 0.390nMAssay Description:Displacement of [125 I] CCK-8 from Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50280834(1-((S)-5-Cyclohexyl-1-methyl-2-oxo-2,3-dihydro-1H-...)
Affinity DataIC50: 0.455nMAssay Description:In vitro test for inhibition of [125I]CCK binding to Cholecystokinin type A receptor from rat pancreatic tissues was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50154434((S)-2-((4S,5S)-2-Benzyl-4-methyl-1,3-dioxo-octahyd...)
Affinity DataIC50: 0.470nMAssay Description:Inhibition of [3H]-pCCK-8 binding to Cholecystokinin type A receptor of rat pancreas homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of [125I](BH)-CCK-8 binding to cholecystokinin type A receptor in rat pancreatic acini; InactiveMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.520nMAssay Description:Inhibition of [3H]pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50369325(CHEMBL1791005)
Affinity DataKi:  0.530nMAssay Description:Binding affinity for Cholecystokinin type A receptor using [125I]BH-CCK-8 in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50170764([(S)-2-(1H-Indol-3-yl)-1-((4aS,5R)-2-naphthalen-1-...)
Affinity DataIC50: 0.590nMAssay Description:Inhibition of 71 pM [125I]BH-(Thr,Nle)CCK-9 binding to rat cholecystokinin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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