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Report error Found 635 for UniProtKB: P30553
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(CHEMBL115121 | YM022 Racemate | YM022 | 1-[(R)-2-O...)
Affinity DataKi:  0.0680nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50286892(1-[(R)-1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pheny...)
Affinity DataIC50: 0.0700nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.0970nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50286884(1-{1-[2-(1-Methyl-cyclopentyl)-2-oxo-ethyl]-2-oxo-...)
Affinity DataIC50: 0.100nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056102(YF-476 | 1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo...)
Affinity DataIC50: 0.100nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(CHEMBL115121 | YM022 Racemate | YM022 | 1-[(R)-2-O...)
Affinity DataIC50: 0.110nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056103(1-(3-Diethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-2...)
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(CHEMBL115121 | YM022 Racemate | YM022 | 1-[(R)-2-O...)
Affinity DataIC50: 0.110nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]CCK-8 as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056099(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-pyridi...)
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056093(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(CHEMBL115121 | YM022 Racemate | YM022 | 1-[(R)-2-O...)
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(CHEMBL115121 | YM022 Racemate | YM022 | 1-[(R)-2-O...)
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50286903(1-[1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pyridin-2...)
Affinity DataIC50: 0.120nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]CCK-8 as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50286897(1-[2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-pyridin-2-yl-...)
Affinity DataIC50: 0.130nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]CCK-8 as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056092(1-(3-Diethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-2...)
Affinity DataIC50: 0.140nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056091(1-[1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl-2,3...)
Affinity DataIC50: 0.160nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM82235(Gastrin I | Gastrin-17 | Gastrin-I-(1-17))
Affinity DataEC50:  0.170nMAssay Description:Agonist activity at gastrin receptor in rat AR4-2J cells assessed as intracellular calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056089(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)
Affinity DataIC50: 0.170nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056095(1-(3-Dimethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-...)
Affinity DataIC50: 0.200nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056098(1-(3-Dimethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-...)
Affinity DataIC50: 0.210nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50286882(1-[(S)-1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pheny...)
Affinity DataIC50: 0.230nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50286882(1-[(S)-1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pheny...)
Affinity DataIC50: 0.230nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]CCK-8 as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50288462((R)-2-{(2R,5S)-2-[(R)-3-((R)-2-Carboxy-pyrrolidine...)
Affinity DataIC50: 0.25nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50348753(CHEMBL1806528)
Affinity DataEC50:  0.270nMAssay Description:Agonist activity at gastrin receptor in rat AR4-2J cells assessed as intracellular calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50286886(1-[1-(3-Cyclohexyl-2-oxo-propyl)-2-oxo-5-phenyl-2,...)
Affinity DataIC50: 0.280nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50092393(3-(2-{[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-su...)
Affinity DataKi:  0.310nMAssay Description:Compound was tested for binding affinity against Cholecystokinin type B receptor expressed in CHO cells on the rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50348752(CHEMBL1807150)
Affinity DataEC50:  0.330nMAssay Description:Agonist activity at gastrin receptor in rat AR4-2J cells assessed as intracellular calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataKi:  0.330nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2011
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50286888(1-{1-[2-(1-Methyl-cyclohexyl)-2-oxo-ethyl]-2-oxo-5...)
Affinity DataIC50: 0.380nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50092405((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-((S)-2-{[...)
Affinity DataEC50:  0.400nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50084033(CHEMBL333994 | FK480 | 1H-Indole-2-carboxylic acid...)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50286891(1-[1-(2-Cyclohexyl-2-oxo-ethyl)-2-oxo-5-phenyl-2,3...)
Affinity DataIC50: 0.400nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50348756(CHEMBL1806532)
Affinity DataEC50:  0.410nMAssay Description:Agonist activity at gastrin receptor in rat AR4-2J cells assessed as intracellular calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.410nMAssay Description:Binding affinity towards Cholecystokinin type B receptor in rat cortex synaptosomes using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.410nMAssay Description:Binding affinity for Cholecystokinin type B receptor using [125I]-BH-CCK-8 in rat cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50286885(1-{1-[2-(1-Methyl-cyclopropyl)-2-oxo-ethyl]-2-oxo-...)
Affinity DataIC50: 0.410nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataKi:  0.420nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056086(1-(3-Amino-phenyl)-3-[(R)-1-(3,3-dimethyl-2-oxo-bu...)
Affinity DataIC50: 0.430nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50024321(CHEMBL1328 | Peptavlon | ICI-50123 | 3-{2-[2-(3-te...)
Affinity DataEC50:  0.430nMAssay Description:Agonist activity at rat CCK2R expressed in rat AR42J cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056096(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-pyridi...)
Affinity DataIC50: 0.440nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]CCK-8 as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056096(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-pyridi...)
Affinity DataIC50: 0.440nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056094(1-(3-Amino-phenyl)-3-[(R)-1-(3,3-dimethyl-2-oxo-bu...)
Affinity DataIC50: 0.5nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056097(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)
Affinity DataIC50: 0.520nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056097(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)
Affinity DataIC50: 0.520nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]CCK-8 as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056097(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)
Affinity DataIC50: 0.520nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataKi:  0.540nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50092408(N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2-{[3-(1H-indol-...)
Affinity DataEC50:  0.560nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50286883(1-[1-(3,3-Dimethyl-2-oxo-pentyl)-2-oxo-5-phenyl-2,...)
Affinity DataIC50: 0.570nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM82304(CAS_122077 | NSC_122077 | SR 27897)
Affinity DataKi:  0.580nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2011
Entry Details Article
PubMed
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