Compile Data Set for Download or QSAR
Report error Found 193 of affinity data for UniProtKB/TrEMBL: P42260
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053067BDBM50053067((2S,3S,4S)-3-Carboxymethyl-4-(1-phenyl-vinyl)-pyrr...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053071BDBM50053071((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-fluoro-3-methyl...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053075BDBM50053075((2S,3S,4S)-4-(1-Biphenyl-3-yl-vinyl)-3-carboxymeth...)
Affinity DataKi:  2.10nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053083BDBM50053083((2S,3S,4S)-3-Carboxymethyl-4-(1-m-tolyl-vinyl)-pyr...)
Affinity DataKi:  2.20nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053080BDBM50053080((2S,3S,4S)-3-Carboxymethyl-4-[1-(3,4-dimethyl-phen...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053088BDBM50053088((2S,3S,4S)-3-Carboxymethyl-4-(1-p-tolyl-vinyl)-pyr...)
Affinity DataKi:  2.60nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053087BDBM50053087((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-fluoro-phenyl)-...)
Affinity DataKi:  2.70nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053064BDBM50053064((2S,3S,4S)-4-[1-(4-Butoxy-phenyl)-vinyl]-3-carboxy...)
Affinity DataKi:  2.80nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053063BDBM50053063((2S,3S,4S)-3-Carboxymethyl-4-[1-(3-methoxy-phenyl)...)
Affinity DataKi:  3.5nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053068BDBM50053068((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-isopropenyl-phe...)
Affinity DataKi:  3.60nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053059BDBM50053059((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-propyl-phenyl)-...)
Affinity DataKi:  3.60nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50002369BDBM50002369(Digensaeure | (3S,4R)-3-(carboxymethyl)-4-(prop-1-...)
Affinity DataKi:  3.70nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053073BDBM50053073((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-methoxy-phenyl)...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053061BDBM50053061((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-chloro-phenyl)-...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053082BDBM50053082((2S,3S,4S)-4-[1-(4-Butyl-phenyl)-vinyl]-3-carboxym...)
Affinity DataKi:  4.80nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252103BDBM50252103(CHEMBL482097 | (2S,3S,4S)-2-CARBOXY-4-[(1Z,3E,5R)-...)
Affinity DataKi:  6.04nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR6More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053065BDBM50053065((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-phenethyloxy-ph...)
Affinity DataKi:  6.20nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053089BDBM50053089((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-ethyl-phenyl)-v...)
Affinity DataKi:  7.70nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053070BDBM50053070((2S,3S,4S)-3-Carboxymethyl-4-{1-[4-(1-methylene-pr...)
Affinity DataKi:  9nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053076BDBM50053076((2S,3S,4S)-4-(1-Biphenyl-4-yl-vinyl)-3-carboxymeth...)
Affinity DataKi:  9.10nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053062BDBM50053062((2S,3S,4S)-3-Carboxymethyl-4-[1-(3,5-dimethyl-phen...)
Affinity DataKi:  9.5nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053074BDBM50053074((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-phenoxy-phenyl)...)
Affinity DataKi:  11.9nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50002369BDBM50002369(Digensaeure | (3S,4R)-3-(carboxymethyl)-4-(prop-1-...)
Affinity DataKi:  12.7nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR6More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50002369BDBM50002369(Digensaeure | (3S,4R)-3-(carboxymethyl)-4-(prop-1-...)
Affinity DataKi:  12.7nMAssay Description:Displacement of [3H]kainic acid from rat recombinant iGluR6(V,C,R) receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053077BDBM50053077((2S,3S,4S)-3-Carboxymethyl-4-[1-(3-phenethyloxy-ph...)
Affinity DataKi:  16nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031704BDBM50031704(2-Amino-4-methyl-pentanedioic acid | (2S,4R)-2-ami...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR6More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053060BDBM50053060((2S,3S,4S)-4-[1-(4-tert-Butyl-phenyl)-vinyl]-3-car...)
Affinity DataKi:  18.5nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50166288BDBM50166288((S)-2-Amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]KA from rat recombinant GluR6 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053079BDBM50053079((2S,3S,4S)-4-[1-(3-Butoxy-phenyl)-vinyl]-3-carboxy...)
Affinity DataKi:  23.3nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50002369BDBM50002369(Digensaeure | (3S,4R)-3-(carboxymethyl)-4-(prop-1-...)
Affinity DataKd:  39nMAssay Description:Displacement of [3H]kainate from rat GLUK6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50211399BDBM50211399((RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazo...)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]KA from rat recombinant GluR6 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50166286BDBM50166286((RS)-2-amino-3-[3-hydroxy-5-(2-ethyl-2H-5-tetrazol...)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]KA from rat recombinant GluR6 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50166285BDBM50166285((RS)-2-amino-3-[3-hydroxy-5-(2-propyl-2H-5-tetrazo...)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]KA from rat recombinant GluR6 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50166287BDBM50166287((RS)-2-amino-3-[3-hydroxy-5-(2-isopropyl-2H-5-tetr...)
Affinity DataKi: >100nMAssay Description:Displacement of [3H]KA from rat recombinant GluR6 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50252051BDBM50252051((2S,4R)-2-amino-4-(3-(methylamino)-3-oxopropyl)pen...)
Affinity DataKi:  123nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR6More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053066BDBM50053066((2S,3S,4S)-3-Carboxymethyl-4-{1-[4-(5-phenyl-penty...)
Affinity DataKi:  126nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 17660BDBM17660(2-amino-3-(3,5-dioxo[1,2,4]oxadiazolidin-2-yl)prop...)
Affinity DataKi:  134nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR6More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053078BDBM50053078((2S,3S,4S)-3-Carboxymethyl-4-{1-[3-(3,3-diphenyl-p...)
Affinity DataKi:  210nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053069BDBM50053069((2S,3S,4R)-3-Carboxymethyl-4-(1-phenyl-vinyl)-pyrr...)
Affinity DataKi:  230nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 17657BDBM17657(L-Glutamic acid | L-Glu | (2S)-2-aminopentanedioic...)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]SYM2081 from rat iGluR6 receptor expressed in Sf9 cells baculovirus system after 1 to 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 17657BDBM17657(L-Glutamic acid | L-Glu | (2S)-2-aminopentanedioic...)
Affinity DataKi:  331nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR6More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 17657BDBM17657(L-Glutamic acid | L-Glu | (2S)-2-aminopentanedioic...)
Affinity DataKi:  331nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluKK2(VCR) receptor expressed in sf9 cells by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 17657BDBM17657(L-Glutamic acid | L-Glu | (2S)-2-aminopentanedioic...)
Affinity DataKi:  332nMAssay Description:Displacement of [3H]kainic acid from rat recombinant iGluR6(V,C,R) receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50426290BDBM50426290(CHEMBL2312682)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluKK2(VCR) receptor expressed in sf9 cells by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50426285BDBM50426285(CHEMBL2312403)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluKK2(VCR) receptor expressed in sf9 cells by liquid scintillati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50002370BDBM50002370((RS)-2-amino-3-(3-hydroxy-5-methylisoxazol-4-yl)-p...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]KA from rat recombinant GluR6 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50185321BDBM50185321(7-nitro-2,3-dioxo-2,3-dihydroquinoxaline-6-carboni...)
Affinity DataKi:  1.05E+3nMAssay Description:Displacement of [3H]kainate from rat GLUK6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50185321BDBM50185321(7-nitro-2,3-dioxo-2,3-dihydroquinoxaline-6-carboni...)
Affinity DataKi:  1.05E+3nMAssay Description:Displacement of [3H]kainate from rat GLUK6 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50002369BDBM50002369(Digensaeure | (3S,4R)-3-(carboxymethyl)-4-(prop-1-...)
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at rat recombinant GluR6(Q) RNA-edited isoform expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, kainate 2(Rat)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50646125BDBM50646125(CHEMBL5595349)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of [3H]-KA from rat GluK2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
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